SCHEMBL20333384

SCHEMBL20333384

COC(Cc1ccc(NC(C)=O)cc1)(C(=O)O)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.50
PTPN1 P18031 1/20 0.48
TSHR P16473 2/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NAPRT Q6XQN6 1/20 0.46
HSD17B10 Q99714 1/20 0.46
KMT2A Q03164 5/20 0.45
MEN1 O00255 4/20 0.45
TDP1 Q9NUW8 2/20 0.45
HPGD P15428 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
MAPT P10636 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
POLB P06746 1/20 0.45
ALDH1A1 P00352 2/20 0.44
CA12 O43570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20347415 0.85 PTPN1 (0.46) SMN1; SMN2PTPN1TSHRHTTL3MBTL1
SCHEMBL20350802 0.84 PTPN1 (0.44) SMN1; SMN2PTPN1TSHRHTTL3MBTL1
SCHEMBL934104 0.78 SMN1; SMN2 (0.52) SMN1; SMN2PTPN1TSHRLMNACYP1A2
SCHEMBL20333383 0.77 MAPT (0.60) SMN1; SMN2TSHRKMT2AMEN1LMNA
SCHEMBL20333381 0.77 RXRA (0.39) SMN1; SMN2PTPN1LMNAALDH1A1CYP3A4
SCHEMBL20350718 0.77 ALDH1A1 (0.50) SMN1; SMN2TSHRL3MBTL1KMT2AMEN1
SCHEMBL11989506 0.76 SMN1; SMN2 (0.55) SMN1; SMN2PTPN1TSHRHTTL3MBTL1
SCHEMBL15577125 0.74 BLM (0.40) SMN1; SMN2PTPN1TSHRHSD17B10KMT2A
SCHEMBL15577140 0.74 BLM (0.40) SMN1; SMN2PTPN1TSHRHSD17B10KMT2A
SCHEMBL20333769 0.74 FFAR1 (0.50) L3MBTL1LMNACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018119284-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF CALITHERA BIOSCIENCES, INC. (US) 2018-06-28 WO disclosed