SCHEMBL20334886

SCHEMBL20334886

O=C(CCl)N(c1ccccc1)c1c[nH]c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 1.00
RAB9A P51151 7/20 1.00
ALDH1A1 P00352 7/20 1.00
KMT2A Q03164 4/20 1.00
MEN1 O00255 3/20 1.00
MITF O75030 2/20 1.00
TDP1 Q9NUW8 1/20 1.00
NPSR1 Q6W5P4 7/20 0.82
MAPT P10636 6/20 0.82
HTT P42858 3/20 0.82
LMNA P02545 2/20 0.82
POLB P06746 1/20 0.58
HKDC1 Q2TB90 1/20 0.54
KDM4E B2RXH2 3/20 0.51
PAX8 Q06710 2/20 0.51
ADAM17 P78536 1/20 0.44
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
S1PR4 O95977 2/20 0.43
S1PR1 P21453 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23094166 0.91 NPC1 (1.00) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL13504941 0.89 NPC1 (0.81) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL12652713 0.89 NPC1 (0.81) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL13475466 0.82 ALDH1A1 (0.70) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL7893567 0.80 MEN1 (0.67) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL21467691 0.80 MAPT (0.81) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL10991862 0.79 ALDH1A1 (0.65) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL7334283 0.77 ALDH1A1 (0.62) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL7343483 0.76 ALDH1A1 (0.61) NPC1RAB9AALDH1A1KMT2AMEN1
SCHEMBL2345303 0.76 ALDH1A1 (1.00) NPC1RAB9AALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10947188-B2 Small molecule ferroptosis inducers THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2021-03-16 US disclosed
US-20190315681-A1 SMALL MOLECULE FERROPTOSIS INDUCERS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2019-10-17 US disclosed
WO-2018118711-A1 SMALL MOLECULE FERROPTOSIS INDUCERS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10947188-B2 Small molecule ferroptosis inducers GPX4, AIFM2, GPX1 NPC1 365/4885RAB9A 2758/4885ALDH1A1 845/4885
US-20190315681-A1 SMALL MOLECULE FERROPTOSIS INDUCERS GPX4, AIFM2, GPX1 NPC1 365/4885RAB9A 2758/4885ALDH1A1 845/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.