SCHEMBL2037498

SCHEMBL2037498

Cc1ccc(-n2nnc(-c3cncs3)n2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 14/20 0.43
NPC1 O15118 13/20 0.43
PKM P14618 3/20 0.43
RECQL P46063 1/20 0.43
MAPT P10636 6/20 0.41
CHRNB2 P17787 2/20 0.40
CHRNA5 P30532 2/20 0.40
CHRNA4 P43681 2/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
NFKB1 P19838 1/20 0.39
CASP3 P42574 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2037353 0.83 RAB9A (0.43) RAB9ANPC1PKMRECQLMAPT
SCHEMBL2037831 0.80 CHRNB2 (0.64) RAB9ANPC1PKMMAPTCHRNB2
SCHEMBL2040546 0.80 RAB9A (0.43) RAB9ANPC1PKMRECQLMAPT
SCHEMBL2039061 0.75 CHRNB2 (0.74) RAB9ANPC1MAPTCHRNB2CHRNA5
SCHEMBL2036415 0.72 CHRNB2 (0.74) RAB9ANPC1PKMMAPTCHRNB2
SCHEMBL13745367 0.71 DYRK1A (0.46) RAB9ANPC1PKMMAPT
SCHEMBL2037773 0.70 NPC1 (0.38) RAB9ANPC1PKMMAPTCHRNB2
SCHEMBL17145305 0.66 SMN1; SMN2 (0.46) KMT2AL3MBTL1MEN1
SCHEMBL4853177 0.64 PTGS1 (0.38) MAPT
SCHEMBL4699663 0.64 GRM5 (0.63) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073298-A1 TETRAZOLE DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 2011-06-23 WO claimed
WO-2011073298-A1 TETRAZOLE DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 2011-06-23 WO disclosed