SCHEMBL2037579

SCHEMBL2037579

Fc1ccc(-n2nnc(-c3ccns3)n2)cn1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 14/20 0.42
NPC1 O15118 13/20 0.42
PKM P14618 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 6/20 0.40
KDM4E B2RXH2 4/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA5 P30532 1/20 0.37
CHRNA4 P43681 1/20 0.37
RECQL P46063 2/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 2/20 0.34
NFKB1 P19838 1/20 0.33
CASP3 P42574 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
GRM5 P41594 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2040546 0.84 RAB9A (0.43) RAB9ANPC1PKMKMT2AMAPT
SCHEMBL2037353 0.80 RAB9A (0.43) RAB9ANPC1PKMKMT2AMAPT
SCHEMBL2036940 0.78 CHRNB2 (0.62) RAB9ANPC1PKMMAPTCHRNB2
SCHEMBL2036408 0.77 NPC1 (0.41) RAB9ANPC1PKMKMT2ACHRNB2
SCHEMBL2041201 0.73 RAB9A (0.59) RAB9ANPC1PKMMAPTKDM4E
SCHEMBL2040507 0.73 NPC1 (0.73) RAB9ANPC1MAPTKDM4ECHRNB2
SCHEMBL2034759 0.70 NPC1 (0.51) RAB9ANPC1PKMKMT2AMAPT
SCHEMBL2036752 0.68 NPC1 (0.46) RAB9ANPC1PKMKMT2AMAPT
SCHEMBL2039666 0.68 NPC1 (0.46) RAB9ANPC1KMT2AMAPTKDM4E
SCHEMBL2033604 0.68 CHRNB2 (0.72) RAB9ANPC1MAPTCHRNB2CHRNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073298-A1 TETRAZOLE DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 2011-06-23 WO claimed
WO-2011073298-A1 TETRAZOLE DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 2011-06-23 WO disclosed