SCHEMBL20384352

SCHEMBL20384352

N#CCSc1ccc(F)c(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.43
MAOB P27338 7/20 0.35
MAOA P21397 5/20 0.35
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.31
KDM4E B2RXH2 1/20 0.31
DAO P14920 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8529340 0.79 ALOX15 (0.41) IDO1MAOBMAOAMEN1ALDH1A1
SCHEMBL20384525 0.78 EPAS1 (0.46) MAOBMAOARXFP1TDP1ALDH1A1
SCHEMBL15067807 0.76 IDO1 (0.40) IDO1MAOACYP1A2CYP2D6CYP2C9
SCHEMBL8528307 0.75 CYP19A1 (0.42) MAOBMAOADAO
SCHEMBL20442961 0.73 KDM4E (0.32) KDM4E
SCHEMBL7952409 0.72 MAOA (0.52) MAOBMAOACYP1A2NPSR1RXFP1
SCHEMBL20384329 0.72 KDM4E (0.38) IDO1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL23340738 0.71 RXFP1 (0.46) MAOBMAOACYP1A2CYP2C9CYP2C19
SCHEMBL16005244 0.70 HTR2A (0.36) IDO1RXFP1KDM4EMEN1ALDH1A1
SCHEMBL6816553 0.70 MAOA (0.50) MAOBMAOANPSR1RXFP1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167939-B Pyrrolo [2,3-c ] pyridine derivatives, preparation method and medical application thereof 江苏豪森药业集团有限公司 2021-12-31 CN disclosed
CN-110198941-B Pyrrolopyridine N-oxide derivative and preparation method and application thereof 江苏豪森药业集团有限公司 2021-09-28 CN disclosed
WO-2018137655-A1 PYRROLO-PYRIDINES N-OXIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-08-02 WO disclosed
WO-2018130174-A1 PYRROLO[2,3-C]PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF IN MEDICINE 江苏豪森药业集团有限公司 2018-07-19 WO disclosed