SCHEMBL8529340

SCHEMBL8529340

N#CCSc1ccc(O)c(Br)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.41
MAOB P27338 4/20 0.35
KMT2A Q03164 3/20 0.34
PKM P14618 1/20 0.34
PTP4A3 O75365 1/20 0.33
PTP4A1 Q93096 1/20 0.33
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
CA14 Q9ULX7 1/20 0.33
CYP19A1 P11511 6/20 0.32
MAOA P21397 2/20 0.32
ALOX12 P18054 1/20 0.32
MEN1 O00255 2/20 0.32
ALDH1A1 P00352 1/20 0.32
IDO1 P14902 1/20 0.31
CA4 P22748 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8746024 0.79 CYP19A1 (0.32) MAOBCYP19A1MAOATTRALB
SCHEMBL8528307 0.79 CYP19A1 (0.42) MAOBCYP19A1MAOA
SCHEMBL20384352 0.79 IDO1 (0.43) MAOBKMT2AMAOAMEN1ALDH1A1
SCHEMBL8526638 0.79 CYP19A1 (0.44) MAOBKMT2ACA1CA2CYP19A1
SCHEMBL9360204 0.76 TSHR (0.36) ALOX15MAOBKMT2APKMMAOA
SCHEMBL5634830 0.76 ALOX15 (0.45) ALOX15MAOBKMT2APKMPTP4A3
SCHEMBL5178452 0.72 NR1H2 (0.44) ALOX15KMT2ACA12CA1CA2
SCHEMBL70601 0.72 ALOX15 (0.54) ALOX15MAOBKMT2ACYP19A1MAOA
SCHEMBL6816553 0.70 MAOA (0.50) MAOBKMT2ACA1CA2CA9
SCHEMBL11589995 0.70 MAOB (0.50) ALOX15MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0692033-B1 ENHANCEMENT OF CHEMILUMINESCENT REACTIONS BRITISH TECH GROUP (GB) 1998-03-11 EP claimed
EP-0505198-B1 A method of enhancing a luminescent reaction, luminometric assay and kits for use in the same SANYO CHEMICAL IND LTD (JP) 1997-01-02 EP claimed
US-5512451-A MIXTURE OF A AROMATIC DIACYL CYCLIC HYDRAZIDE, PEROXIDASE CATALYST AND OXIDIZER BRITISH TECHNOLOGY GROUP LIMITED (GB) 1996-04-30 US claimed
EP-0692033-A1 ENHANCEMENT OF CHEMILUMINESCENT REACTIONS BTG INTERNATIONAL LIMITED (GB) 1996-01-17 EP claimed
WO-1994023060-A2 ENHANCEMENT OF CHEMILUMINESCENT REACTIONS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1994-10-13 WO claimed
EP-0505198-A1 A method of enhancing a luminescent reaction, luminometric assay and kits for use in the same SANYO CHEMICAL INDUSTRIES, LTD. (JP) 1992-09-23 EP claimed
EP-0692033-B1 ENHANCEMENT OF CHEMILUMINESCENT REACTIONS BRITISH TECH GROUP (GB) 1998-03-11 EP disclosed
EP-0505198-B1 A method of enhancing a luminescent reaction, luminometric assay and kits for use in the same SANYO CHEMICAL IND LTD (JP) 1997-01-02 EP disclosed
US-5512451-A MIXTURE OF A AROMATIC DIACYL CYCLIC HYDRAZIDE, PEROXIDASE CATALYST AND OXIDIZER BRITISH TECHNOLOGY GROUP LIMITED (GB) 1996-04-30 US disclosed
EP-0692033-A1 ENHANCEMENT OF CHEMILUMINESCENT REACTIONS BTG INTERNATIONAL LIMITED (GB) 1996-01-17 EP disclosed
US-5424194-A Chemiluminescence SANYO CHEMICAL INDUSTRIES, LTD. (JP) 1995-06-13 US disclosed
WO-1994023060-A2 ENHANCEMENT OF CHEMILUMINESCENT REACTIONS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1994-10-13 WO disclosed
EP-0505198-A1 A method of enhancing a luminescent reaction, luminometric assay and kits for use in the same SANYO CHEMICAL INDUSTRIES, LTD. (JP) 1992-09-23 EP disclosed