SCHEMBL20418643

SCHEMBL20418643

CN(C(=O)C(F)(F)F)c1ccc(C(=O)OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.44
GRM5 P41594 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KEAP1 Q14145 2/20 0.41
NFE2L2 Q16236 2/20 0.41
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20418657 0.81 RAB9A (0.43) ALDH1A1MAPTHPGDHTTL3MBTL1
SCHEMBL29447544 0.81 RAB9A (0.43) ALDH1A1MAPTHPGDHTTL3MBTL1
SCHEMBL20418653 0.80 ALDH1A1 (0.44) ALDH1A1TDP1CYP3A4TSHRMAPK1
SCHEMBL20401096 0.79 TSPO (0.40) ALDH1A1MAPTHPGDHTTTDP1
SCHEMBL19667309 0.78 HTT (0.48) ALDH1A1HTTTDP1CYP3A4TSHR
SCHEMBL20418711 0.78 HTT (0.36) ALDH1A1HTTTDP1TSHRKEAP1
SCHEMBL29447580 0.78 HTT (0.36) ALDH1A1HTTTDP1TSHRKEAP1
SCHEMBL29447455 0.77 KEAP1 (0.37) ALDH1A1HTTKEAP1NFE2L2
SCHEMBL8677521 0.77 MTNR1B (0.44) ALDH1A1MAPTHPGDGRM5TDP1
SCHEMBL20418487 0.76 HTR2C (0.46) ALDH1A1MAPTHPGDHTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018136935-A1 2-ARYLSULFONAMIDO-N-ARYLACETAMIDE DERIVATIZED STAT3 INHIBITORS UNIVERSITY OF HAWAII (US) 2018-07-26 WO disclosed