SCHEMBL20459575

SCHEMBL20459575

Cc1nc(Cl)cc(NC(c2ccccc2)(c2ccccc2)c2ccccc2)c1C(=N)N1CCOCC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
CNR1 P21554 1/20 0.36
LRRK2 Q5S007 5/20 0.35
HPGD P15428 3/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPK1 P28482 1/20 0.35
TSHR P16473 2/20 0.34
EPAS1 Q99814 1/20 0.34
USP2 O75604 2/20 0.34
F10 P00742 1/20 0.34
KDM4E B2RXH2 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20459834 0.86 SMN1; SMN2 (0.33) SMN1; SMN2LRRK2HPGDALDH1A1TSHR
SCHEMBL20459560 0.85 SMN1; SMN2 (0.35) SMN1; SMN2HPGDALDH1A1TSHRUSP2
SCHEMBL20459591 0.68 TACR1 (0.31) KDM4E
SCHEMBL883641 0.63 PIK3CA (0.47) SMN1; SMN2LRRK2ALDH1A1
SCHEMBL23617989 0.59 TSHR (0.56) SMN1; SMN2HPGDALDH1A1TSHRUSP2
SCHEMBL17108576 0.59 VNN1 (0.34) F10
SCHEMBL926070 0.59 KCNN4 (0.35) ALDH1A1TSHR
SCHEMBL20459751 0.59 VNN1 (0.37) SMN1; SMN2
SCHEMBL24975805 0.59 LMNA (0.47) SMN1; SMN2HPGDALDH1A1TSHRF10
SCHEMBL7746677 0.58 ALDH1A1 (0.71) SMN1; SMN2CNR1HPGDALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900241-B1 NOVEL COMPOUNDS THAT ARE ERK INHIBITORS MERCK SHARP & DOHME (US) 2018-08-08 EP disclosed