SCHEMBL20459591

SCHEMBL20459591

CC(=N)c1c(NC(c2ccccc2)(c2ccccc2)c2ccccc2)cc(Cl)nc1CO

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.31
KDM4E B2RXH2 1/20 0.30
CTSA P10619 1/20 0.30
VNN1 O95497 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20459834 0.80 SMN1; SMN2 (0.33) KDM4E
SCHEMBL20459575 0.68 SMN1; SMN2 (0.37) KDM4E
SCHEMBL926070 0.67 KCNN4 (0.35) VNN1
SCHEMBL20018530 0.67 VNN1 (0.33) VNN1
SCHEMBL20459545 0.65 KCNN4 (0.35) VNN1
SCHEMBL17108576 0.64 VNN1 (0.34) VNN1
SCHEMBL20459751 0.63 VNN1 (0.37) VNN1
SCHEMBL19671830 0.60 ALDH1A1 (0.46) KDM4E
SCHEMBL11721973 0.60 KCNN4 (0.50)
SCHEMBL19672008 0.59 KCNK2 (0.34) VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900241-B1 NOVEL COMPOUNDS THAT ARE ERK INHIBITORS MERCK SHARP & DOHME (US) 2018-08-08 EP disclosed