Bromide

Bromide

SCHEMBL20501902

Br.Br.NCCCCCNC1(c2ccccc2)CCCCC1

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2A known ✓ Q12879 2/20 0.97
GRIN2D O15399 2/20 0.97
GRIN3B O60391 2/20 0.97
GRIA1 P42261 2/20 0.97
GRIA2 P42262 2/20 0.97
GRIA3 P42263 2/20 0.97
GRIA4 P48058 2/20 0.97
GRIN1 Q05586 2/20 0.97
GRIN2B Q13224 2/20 0.97
GRIN2C Q14957 2/20 0.97
GRIN3A Q8TCU5 2/20 0.97
DPP4 P27487 1/20 0.41
KDM1A O60341 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19242786 0.98 GRIN2D (1.00) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL19242764 0.97 GRIN2D (0.97) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL19242714 0.84 GRIN2D (0.74) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9765029 0.81 GRIN2D (0.70) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL23068594 0.80 GRIN2D (0.68) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL5328724 0.80 GRIN2D (0.68) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL30151574 0.79 GRIN2D (0.67) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL19242654 0.79 GRIN2D (0.67) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL1261302 0.78 GRIN2D (0.65) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL29604371 0.76 GRIN2D (0.62) GRIN2DGRIN3BGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12616807-B2 Medical counter measures including dry powder formulations and associated methods Belhaven BioPharma Inc. (US) 2026-05-05 US disclosed
US-12274761-B2 Compositions and methods to detect GLUA1 in brain and to identify the presence of GLUA1-mediated PTSD NEUROVATION LABS, INC. (US) 2025-04-15 US disclosed
US-20240299680-A1 MEDICAL COUNTER MEASURES INCLUDING DRY POWDER FORMULATIONS AND ASSOCIATED METHODS Belhaven BioPharma Inc. (US) 2024-09-12 US disclosed
US-12005185-B2 Medical counter measures including dry powder formulations and associated methods Belhaven BioPharma Inc. (US) 2024-06-11 US disclosed
US-20230191047-A1 MEDICAL COUNTER MEASURES INCLUDING DRY POWDER FORMULATIONS AND ASSOCIATED METHODS Belhaven BioPharma Inc. (US) 2023-06-22 US disclosed
WO-2023114462-A1 MEDICAL COUNTER MEASURES INCLUDING DRY POWDER FORMULATIONS AND ASSOCIATED METHODS Belhaven BioPharma Inc. (US) 2023-06-22 WO disclosed
US-11439715-B2 Compositions and methods to detect GLUA1 in brain and to identify the presence of GLUA1-mediated post-traumatic stress disorder and other neurological disorders NEUROVATION LABS, INC. (US) 2022-09-13 US disclosed
US-20220125956-A1 COMPOSITIONS AND METHODS TO DETECT GLUA1 IN BRAIN AND TO IDENTIFY THE PRESENCE OF GLUA1-MEDIATED PTSD NEUROVATION LABS, INC. 2022-04-28 US disclosed
US-20210069358-A1 COMPOSITIONS AND METHODS TO DETECT GLUA1 IN BRAIN AND TO IDENTIFY THE PRESENCE OF GLUA1-MEDIATED POST-TRAUMATIC STRESS DISORDER AND OTHER NEUROLOGICAL DISORDERS NEUROVATION LABS INC (US) 2021-03-11 US disclosed
US-20200030304-A1 MITIGATION OF CNS DISORDERS BY COMBINATION THERAPY USING NEUROSTEROIDS, AND AMPA BLOCKERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-01-30 US disclosed
WO-2019046240-A1 COMPOSITIONS AND METHODS TO DETECT GLUA1 IN BRAIN AND TO IDENTIFY GLUA1-MEDIATED POST-TRAUMATIC STRESS DISORDER NEUROVATION LABS, INC. (US) 2019-03-07 WO disclosed
WO-2018169798-A9 MITIGATION OF CNS DISORDERS BY COMBINATION THERAPY USING NEUROSTEROIDS, AND AMPA BLOCKERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-10-18 WO disclosed
WO-2018169798-A1 MITIGATION OF CNS DISORDERS BY COMBINATION THERAPY USING NEUROSTEROIDS, AND AMPA BLOCKERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-09-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200030304-A1 MITIGATION OF CNS DISORDERS BY COMBINATION THERAPY USING NEUROSTEROIDS, AND AMPA BLOCKERS GABRA4, GABRG1, GABRB2 GRIN2A 31/4885GRIN2D 82/4885GRIN3B 51/4885
US-20210069358-A1 COMPOSITIONS AND METHODS TO DETECT GLUA1 IN BRAIN AND TO IDENTIFY THE PRESENCE OF GLUA1-MEDIATED POST-TRAUMATIC STRESS DISORDER AND OTHER NEUROLOGICAL DISORDERS GRIA1, GRIA2, GRIA3 GRIN2A 6/4885GRIN2D 25/4885GRIN3B 19/4885
US-12616807-B2 Medical counter measures including dry powder formulations and associated methods ADRB2, ADRB3, MC5R GRIN2A 568/4885GRIN2D 406/4885GRIN3B 499/4885
US-12274761-B2 Compositions and methods to detect GLUA1 in brain and to identify the presence of GLUA1-mediated PTSD GRIA1, GRIA2, GRIA3 GRIN2A 6/4885GRIN2D 27/4885GRIN3B 15/4885
US-20220125956-A1 COMPOSITIONS AND METHODS TO DETECT GLUA1 IN BRAIN AND TO IDENTIFY THE PRESENCE OF GLUA1-MEDIATED PTSD GRIA1, GRIA2, GRIA3 GRIN2A 6/4885GRIN2D 27/4885GRIN3B 15/4885
US-11439715-B2 Compositions and methods to detect GLUA1 in brain and to identify the presence of GLUA1-mediated post-traumatic stress disorder and other neurological disorders GRIA1, GRIA2, GRIA3 GRIN2A 6/4885GRIN2D 25/4885GRIN3B 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.