SCHEMBL2051089

SCHEMBL2051089

Fc1cccc(-c2ccc[c]c2C(F)(F)F)c1F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.34
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
PDK2 Q15119 2/20 0.31
MPL P40238 1/20 0.30
BCAT1 P54687 1/20 0.30
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2431241 0.85 HTR1A (0.33) HSD11B1GPBAR1PDK2
SCHEMBL2053031 0.84 PDK2 (0.38) GPBAR1PDK2
SCHEMBL15638416 0.83 GPBAR1 (0.36) GPBAR1PDK2MPL
SCHEMBL15637439 0.79 GPR3 (0.33) TRPA1
SCHEMBL81364 0.78
SCHEMBL2053315 0.76 PDK2 (0.35) HSD11B1GPBAR1PDE3BPDE3APDK2
SCHEMBL2049471 0.76 HSD11B1 (0.46) HSD11B1PDE3BPDE3APDK2MPL
SCHEMBL2050765 0.76 PTPN1 (0.36) GPBAR1PDE3BPDE3APDK2
SCHEMBL12815748 0.76 CCNE2 (0.35) HSD11B1CCNE2CCNE1CDK2BCAT1
SCHEMBL1115213 0.74 HSD11B1 (0.36) HSD11B1CCNE2CCNE1CDK2BCAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903440-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer CropScience AG (DE) 2015-08-12 EP disclosed
WO-2014053450-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2014-04-10 WO disclosed
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed