SCHEMBL20523587

SCHEMBL20523587

CCOc1cc(Br)cc(-c2ccccc2NS(C)(=O)=O)c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.46
LMNA P02545 4/20 0.43
PTPN1 P18031 3/20 0.41
PTPN2 P17706 1/20 0.41
PTPN6 P29350 1/20 0.41
ESRRA P11474 1/20 0.40
NR3C1 P04150 2/20 0.40
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
MCL1 Q07820 1/20 0.39
TSHR P16473 2/20 0.39
KDM4E B2RXH2 1/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
PARP14 Q460N5 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
APAF1 O14727 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20523653 0.86 SLC22A12 (0.48) NR3C1ALOX5APFEN1MCL1KDM4E
SCHEMBL20523469 0.73 FYN (0.50) ALOX5APFEN1POLB
SCHEMBL30016133 0.72 PTPN1 (0.54) HSD17B10LMNAPTPN1PTPN2PTPN6
SCHEMBL29134872 0.72 PTPN1 (0.54) HSD17B10LMNAPTPN1PTPN2PTPN6
SCHEMBL20523589 0.71 ALDH1A1 (0.48) LMNAKDM4EALDH1A1MAPT
SCHEMBL20523720 0.67 KMT2A (0.43) KDM4EALDH1A1
SCHEMBL20523546 0.66 NR3C1 (0.41) NR3C1KEAP1NFE2L2ALDH1A1
SCHEMBL4667179 0.64 MCL1 (0.61) LMNAALOX5APFEN1MCL1TSHR
SCHEMBL10094332 0.64 L3MBTL1 (0.74) HSD17B10LMNAALOX5APFEN1MCL1
SCHEMBL13848266 0.63 L3MBTL1 (0.54) NR3C1ALOX5APFEN1MCL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600307-A1 COMPOSITIONS FOR USE IN METHODS OF INHIBITING PROTEIN KINASES University of Houston System (US) 2020-02-05 EP disclosed
WO-2018183633-A1 COMPOSITIONS FOR USE IN METHODS OF INHIBITING PROTEIN KINASES UNIVERSITY OF HOUSTON SYSTEM (US) 2018-10-04 WO disclosed