SCHEMBL2053354

SCHEMBL2053354

Fc1ccc(-c2[c]ccc(C(F)(F)F)c2)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MPL P40238 1/20 0.35
ALOX5AP P20292 4/20 0.34
FEN1 P39748 4/20 0.34
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
GPR3 P46089 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
PDE2A O00408 3/20 0.33
IDO1 P14902 1/20 0.32
APP P05067 2/20 0.31
HSD11B1 P28845 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2052904 0.87 MPL (0.35) MPLALOX5APFEN1GPBAR1CYP1A1
SCHEMBL433493 0.82 ALDH1A1 (0.37) GPR3IDO1ALDH1A1
SCHEMBL2432403 0.81 GPR3 (0.41) MPLGPR3GPBAR1PDE2AHSD11B1
SCHEMBL434555 0.79 CNR1 (0.34) GPR3IDO1ALDH1A1
SCHEMBL1690372 0.77 SMN1; SMN2 (0.34) PDE2A
SCHEMBL925238 0.76 PIK3R1 (0.34) GPR3IDO1ALDH1A1
SCHEMBL2051071 0.76 ALDH1A1 (0.39) GPR3IDO1ALDH1A1
SCHEMBL2049535 0.75 HSD11B1 (0.35) GPR3GPBAR1PDE2AHSD11B1
SCHEMBL28263706 0.75 CES2 (0.38) MPLALOX5APFEN1POLBGPR3
SCHEMBL12076488 0.75 ALOX5AP (0.44) ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed