SCHEMBL2049535

SCHEMBL2049535

Fc1cccc(-c2[c]ccc(C(F)(F)F)c2)c1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.35
CES2 O00748 1/20 0.35
PDE2A O00408 5/20 0.34
PDE10A Q9Y233 3/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
CHRM5 P08912 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
GPR3 P46089 1/20 0.33
P2RX1 P51575 1/20 0.32
P2RX7 Q99572 1/20 0.32
KCNH2 Q12809 1/20 0.32
MGLL Q99685 1/20 0.32
MAT2A P31153 1/20 0.31
PDE6D O43924 1/20 0.31
PDE6A P16499 1/20 0.31
PDE6G P18545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2432403 0.87 GPR3 (0.41) HSD11B1CES2PDE2APDE10AGPBAR1
SCHEMBL2053324 0.81 CES2 (0.38) CES2PDE2ATSHRMAPK1TAAR1
SCHEMBL2017429 0.80 CYP11B1 (0.34) HSD11B1
SCHEMBL8907524 0.80 PIK3R1 (0.33) CES2PDE3BPDE3A
SCHEMBL2053205 0.77 ACHE (0.35) HSD11B1GPR3
SCHEMBL9579904 0.77 SLC9A1 (0.33) CES2
SCHEMBL5778162 0.77 HSD11B1 (0.38) HSD11B1TSHRGPR3
SCHEMBL5323119 0.76 CYP1A1 (0.39) CES2GPR3
SCHEMBL2053354 0.75 MPL (0.35) HSD11B1PDE2AGPBAR1GPR3
SCHEMBL2052904 0.75 MPL (0.35) PDE2APDE10AGPBAR1CHRM5PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed