SCHEMBL2054840

SCHEMBL2054840

BCC(=O)NCCCc1nc2c(OCc3ccc(CNC(C)=O)cc3)nc(N)nc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MGMT P16455 2/20 0.41
PIN1 Q13526 2/20 0.38
MPO P05164 5/20 0.36
MTNR1A P48039 4/20 0.34
MTNR1B P49286 4/20 0.34
TPO P07202 1/20 0.33
CYP3A4 P08684 1/20 0.33
EPX P11678 1/20 0.33
KIF11 P52732 1/20 0.32
ATR Q13535 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
HDAC3 O15379 2/20 0.31
HDAC1 Q13547 2/20 0.31
HDAC2 Q92769 2/20 0.31
HDAC8 Q9BY41 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054847 0.80 CA2 (0.38) MGMTPIN1HDAC3HDAC1HDAC2
SCHEMBL2054825 0.78 HDAC1 (0.43) MGMTPIN1HDAC3HDAC1HDAC2
SCHEMBL2054841 0.78 CA12 (0.51)
SCHEMBL2054842 0.77 PIN1 (0.51) PIN1MPOHDAC1POLBMAPT
SCHEMBL2097032 0.76 CA1 (0.39) PIN1MPOTLR7HDAC1
SCHEMBL2098147 0.76 PIN1 (0.57) MGMTPIN1MPOTPOCYP3A4
SCHEMBL2054844 0.75 L3MBTL1 (0.43) MGMTMPOTPOCYP3A4EPX
SCHEMBL12252403 0.74 MGMT (0.58) MGMTPIN1MPOTPOCYP3A4
SCHEMBL2101048 0.71 PIN1 (0.44) PIN1MPOHDAC3HDAC1HDAC2
SCHEMBL2101045 0.71 PIN1 (0.44) PIN1MPOHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase EPFL ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2007-10-18 US disclosed
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase EPFL ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase AGT, AGXT, AGTR1 MGMT 303/4885PIN1 2756/4885MPO 3210/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.