SCHEMBL20564634

SCHEMBL20564634

O=C(O)NC1CC=C(OS(=O)(=O)C(F)(F)F)CC1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.36
HTR1D P28221 2/20 0.36
DRD3 P35462 2/20 0.36
CXCR2 P25025 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL587951 0.85 BTK (0.40) DRD2HTR1DDRD3
SCHEMBL16843297 0.84 DRD2 (0.38) DRD2HTR1DDRD3
SCHEMBL10280563 0.83 DRD2 (0.37) DRD2HTR1DDRD3
SCHEMBL13354535 0.82 DRD2 (0.33) DRD2HTR1DDRD3
SCHEMBL2481313 0.80 KDM4E (0.43)
SCHEMBL16783722 0.80 ALDH1A1 (0.50)
SCHEMBL12174857 0.80 MAPT (0.34) DRD2HTR1DDRD3CXCR2
SCHEMBL5544919 0.78 RORC (0.34) DRD2HTR1DDRD3CXCR2
SCHEMBL5544926 0.78 RORC (0.34) DRD2HTR1DDRD3CXCR2
SCHEMBL13132554 0.77 DRD2 (0.33) DRD2HTR1DDRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3442973-B1 NOVEL COMPOUNDS AS AUTOTAXIN INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME LEGOCHEM BIOSCIENCES INC (KR) 2022-08-31 EP disclosed
EP-3442973-A1 NOVEL COMPOUNDS AS AUTOTAXIN INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Legochem Bioscience Ltd. (KR) 2019-02-20 EP disclosed
WO-2018212534-A1 NOVEL COMPOUNDS AS AUTOTAXIN INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME LEGOCHEM BIOSCIENCES, INC. (KR) 2018-11-22 WO disclosed