SCHEMBL20573162

SCHEMBL20573162

CCOC(=O)C(C)(C)Cc1cc(Br)ccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP3A4 P08684 2/20 0.38
MAPT P10636 2/20 0.38
CYP2D6 P10635 1/20 0.38
MMP8 P22894 1/20 0.38
ALDH1A1 P00352 7/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
GAA P10253 2/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
LNPEP Q9UIQ6 1/20 0.35
CYP4F2 P78329 2/20 0.35
CYP4A11 Q02928 2/20 0.35
ABCB11 O95342 1/20 0.35
TSHR P16473 1/20 0.35
HTR2A P28223 1/20 0.35
PMP22 Q01453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5140898 0.80 CYP1A2 (0.48) KDM4ECYP1A2MMP8ALDH1A1SMN1; SMN2
SCHEMBL21541959 0.79 SHMT1 (0.42) KDM4ECYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL20669564 0.77 ALDH1A1 (0.39) KDM4ECYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL30163570 0.77 MEN1 (0.44) KDM4EMAPTALDH1A1SMN1; SMN2GAA
SCHEMBL9952026 0.77 MEN1 (0.44) KDM4EMAPTALDH1A1SMN1; SMN2GAA
SCHEMBL24369218 0.75 ALDH1A1 (0.37) KDM4ECYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL31422404 0.75 PPARA (0.47) KDM4ECYP1A2CYP3A4ALDH1A1SMN1; SMN2
SCHEMBL10237568 0.74 RIPK1 (0.50) MAPTMMP8ALDH1A1PPARAL3MBTL1
SCHEMBL17709821 0.74 MMP8 (0.43) KDM4ECYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL16737338 0.74 CYP4F2 (0.45) KDM4ECYP1A2CYP2C19CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3212641-B1 THIAZOLES AS MODULATORS OF RORYT JANSSEN PHARMACEUTICA NV (BE) 2018-12-05 EP disclosed