SCHEMBL20588595

SCHEMBL20588595

CC(=O)NCCNC(=O)Nc1cc(F)c(Oc2ccnc3c2c(Br)cn3COCC[Si](C)(C)C)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 2/20 0.34
TBK1 Q9UHD2 2/20 0.33
ROCK2 O75116 1/20 0.33
OPRK1 P41145 1/20 0.33
MET P08581 6/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MST1R Q04912 4/20 0.32
AXL P30530 2/20 0.32
BRAF P15056 1/20 0.32
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
KIT P10721 1/20 0.32
SRC P12931 1/20 0.32
KDR P35968 1/20 0.32
IDO1 P14902 3/20 0.32
CNR1 P21554 1/20 0.31
ABL1 P00519 1/20 0.31
RET P07949 1/20 0.31
PDGFRB P09619 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20588679 0.93 MET (0.35) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20588354 0.92 TBK1 (0.36) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20588441 0.92 ROCK2 (0.32) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20587523 0.92 MAP4K1 (0.35) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20587612 0.92 ROCK2 (0.33) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20588349 0.91 MAP4K1 (0.35) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20588769 0.91 ROCK2 (0.34) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20587816 0.90 MAP4K1 (0.40) MAP4K1TBK1METBRAFKIT
SCHEMBL20587700 0.90 MAP4K1 (0.36) MAP4K1TBK1ROCK2OPRK1MET
SCHEMBL20587966 0.90 TBK1 (0.35) MAP4K1TBK1ROCK2OPRK1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3638669-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES Bayer Pharma Aktiengesellschaft (DE) 2020-04-22 EP disclosed
WO-2018228920-A1 SUBSTITUTED PYRROLOPYRIDINE-DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-12-20 WO disclosed