SCHEMBL20708552

SCHEMBL20708552

O=CN1CCN(c2cccc(Cl)c2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.60
LMNA P02545 1/20 0.60
MAPT P10636 1/20 0.60
ALOX12 P18054 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
HTR1A P08908 2/20 0.59
HTR2A P28223 2/20 0.59
HTR7 P34969 2/20 0.59
HTR6 P50406 2/20 0.59
HTR3E A5X5Y0 2/20 0.59
HTR3B O95264 2/20 0.59
HTR3A P46098 2/20 0.59
HTR3D Q70Z44 2/20 0.59
HTR3C Q8WXA8 2/20 0.59
TP53 P04637 1/20 0.59
CYP1A2 P05177 1/20 0.59
ADRB1 P08588 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
THRB P10828 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6714846 0.87 ALDH1A1 (0.75) ALDH1A1LMNAMAPTALOX12SMN1; SMN2
SCHEMBL11100857 0.87 ALDH1A1 (0.75) ALDH1A1LMNAMAPTALOX12SMN1; SMN2
SCHEMBL9646111 0.85 ALDH1A1 (0.73) ALDH1A1LMNAMAPTALOX12SMN1; SMN2
SCHEMBL13801242 0.81 CHRM2 (0.53) ALDH1A1LMNAMAPTALOX12SMN1; SMN2
SCHEMBL23222244 0.81 DRD2 (0.56) ALDH1A1LMNAMAPTHTR7
SCHEMBL5698648 0.81 SMN1; SMN2 (0.47) LMNAMAPTSMN1; SMN2CYP1A2CYP3A4
SCHEMBL11889954 0.81 ADRB1 (0.57) ALDH1A1LMNAMAPTSMN1; SMN2HTR7
SCHEMBL4052281 0.81 AKR1C3 (0.52) ALDH1A1LMNAMAPTSMN1; SMN2HTR3E
SCHEMBL27940445 0.80 KCNH2 (0.55) ALDH1A1LMNAMAPTALOX12SMN1; SMN2
SCHEMBL8717879 0.79 AKR1C3 (0.54) ALDH1A1LMNAMAPTSMN1; SMN2HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3237406-B1 5-[(PIPERAZIN-1-YL)-3-OXO-PROPYL]-IMIDAZOLIDINE-2,4-DIONE DERIVATIVES AS ADAMTS INHIBITORS FOR THE TREATMENT OF OSTEOARTHRITIS GALAPAGOS NV (BE) 2019-02-06 EP disclosed
US-9314538-B2 Nucleic acid molecules encoding antibody drug conjugates (ADC) that bind to 191P4D12 proteins AGENSYS, INC. (US) 2016-04-19 US disclosed