SCHEMBL2074286

SCHEMBL2074286

CC(C)(C)[Si](C)(C)OCc1cn(COCC[Si](C)(C)C)cn1

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DUT P33316 1/20 0.35
DGAT1 O75907 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31631922 0.83 DGAT1 (0.33) DGAT1
SCHEMBL14151718 0.82 GRM5 (0.35) DGAT1
SCHEMBL22093251 0.80 DGAT1 (0.34) DGAT1
SCHEMBL5764924 0.79 KDM4E (0.35) DGAT1
SCHEMBL22093263 0.79 CPB1 (0.33) DGAT1
SCHEMBL3841245 0.77 DGAT1 (0.33) DGAT1
SCHEMBL2473549 0.76 DGAT1 (0.34) DGAT1
SCHEMBL13560614 0.75 SMYD2 (0.35) DGAT1
SCHEMBL15613781 0.74 GRM5 (0.32) DGAT1
SCHEMBL18431180 0.74 DGAT1 (0.32) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220388964-A1 (AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS HIBERCELL, INC. 2022-12-08 US disclosed
US-20220388964-A1 (AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS HIBERCELL, INC. 2022-12-08 US disclosed
WO-2020210828-A1 (AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS HIBERCELL, INC. (US) 2020-10-15 WO disclosed
EP-1828171-B1 HETEROCYCLE DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ANGELETTI P IST RICHERCHE BIO (IT) 2014-03-12 EP disclosed
US-8304419-B2 Chemical compounds GLAXOSMITHKLINE LLC (US) 2012-11-06 US disclosed
US-7863294-B2 Heterocycle derivatives as histone deacetylase (HDAC) inhibitors INSTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-01-04 US disclosed
US-7863294-B2 Heterocycle derivatives as histone deacetylase (HDAC) inhibitors INSTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-01-04 US disclosed
US-20090048228-A1 Heterocycle Derivatives As Histone Deacetylase (Hdac) Inhibitors MSD ITALIA S.R.L. (IT) 2009-02-19 US disclosed
US-20090048228-A1 Heterocycle Derivatives As Histone Deacetylase (Hdac) Inhibitors MSD ITALIA S.R.L. (IT) 2009-02-19 US disclosed
US-7081466-B2 2-aroylimidazole compounds for treating cancer SYNTA PHARMACEUTICALS CORP. (US) 2006-07-25 US disclosed
US-20040186129-A1 2-Aroylimidazole compounds for treating cancer KOYA KEIZO (US) 2004-09-23 US disclosed
EP-1427413-A2 2-AROYLIMIDAZOLE COMPOUNDS FOR TREATING CANCER Synta Pharmaceuticals Corporation (US) 2004-06-16 EP disclosed
US-6743919-B2 INCLUDING MULTI-DRUG RESISTANT CANCER CELLS FROM A NUMBER OF DIFFERENT TISSUE TYPES SYNTA PHARMACEUTICALS CORP. 2004-06-01 US disclosed
US-20030096836-A1 2-Aroylimidazole compounds for treating cancer SBR PHARMACEUTICALS CORP. 2003-05-22 US disclosed
WO-2003022274-A2 2-AROYLIMIDAZOLE COMPOUNDS FOR TREATING CANCER SYNTA PHARMACEUTICALS CORP. (US) 2003-03-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048228-A1 Heterocycle Derivatives As Histone Deacetylase (Hdac) Inhibitors HDAC1, HDAC5, HDAC11 DUT 1822/4885DGAT1 2075/4885
US-20030096836-A1 2-Aroylimidazole compounds for treating cancer NR4A1, NR0B2, NR0B1 DUT 155/4885DGAT1 3518/4885
US-20040186129-A1 2-Aroylimidazole compounds for treating cancer TOP2B, HDAC11, CYP4B1 DUT 106/4885DGAT1 3457/4885
US-20220388964-A1 (AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS EIF2AK4, GCN1, GNAI2 DUT 1315/4885DGAT1 1538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.