SCHEMBL20765488

SCHEMBL20765488

Cc1ccc(CN2CCN(C(=O)c3ccc4[nH]c(C)nc4c3)C(C)C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.44
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
PLA2G2A P14555 1/20 0.42
MAPK14 Q16539 1/20 0.41
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CHEK2 O96017 2/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
MGLL Q99685 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
HSD11B1 P28845 1/20 0.38
ROCK2 O75116 2/20 0.38
CCR2 P41597 1/20 0.38
ROCK1 Q13464 1/20 0.38
GHSR Q92847 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20765484 1.00 CCR1 (0.44) CCR1BCHEACHEPLA2G2AMAPK14
SCHEMBL20765824 0.88 BCHE (0.41) BCHEACHECHEK2KDM4EALDH1A1
SCHEMBL20765826 0.88 BCHE (0.41) BCHEACHECHEK2KDM4EALDH1A1
SCHEMBL20765527 0.83 MAPK14 (0.44) BCHEACHEPLA2G2AMAPK14DRD2
SCHEMBL20765524 0.83 MAPK14 (0.44) BCHEACHEPLA2G2AMAPK14DRD2
SCHEMBL20765509 0.82 GHSR (0.47) MAPK14HTTPTGDR2KDM4EALDH1A1
SCHEMBL20765512 0.82 GHSR (0.47) MAPK14HTTPTGDR2KDM4EALDH1A1
SCHEMBL17954168 0.72 ALDH1A1 (0.51) MAPK14L3MBTL1KDM4EALDH1A1POLB
SCHEMBL20765458 0.72 BCHE (0.42) BCHEACHEMAPK14ALDH1A1POLB
SCHEMBL20765490 0.71 MAPK14 (0.54) BCHEACHEMAPK14L3MBTL1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed