SCHEMBL20765509

SCHEMBL20765509

COc1ccccc1CN1CCN(C(=O)c2ccc3[nH]c(C)nc3c2)[C@@H](C)C1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 3/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.45
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
USP2 O75604 2/20 0.41
MAPK1 P28482 1/20 0.41
ROCK2 O75116 1/20 0.41
CYP2D6 P10635 5/20 0.41
CYP3A4 P08684 2/20 0.41
DRD2 P14416 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
DRD3 P35462 1/20 0.41
DRD4 P21917 1/20 0.40
POLB P06746 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20765512 1.00 GHSR (0.47) GHSRPTGDR2ALDH1A1KDM4EHTT
SCHEMBL20782581 0.86 ACHE (0.41) ALDH1A1KDM4EHTTUSP2ROCK2
SCHEMBL20765484 0.82 CCR1 (0.44) GHSRPTGDR2ALDH1A1KDM4EHTT
SCHEMBL20765488 0.82 CCR1 (0.44) GHSRPTGDR2ALDH1A1KDM4EHTT
SCHEMBL20765527 0.80 MAPK14 (0.44) GHSRDRD2MEN1KMT2ADRD3
SCHEMBL20765524 0.80 MAPK14 (0.44) GHSRDRD2MEN1KMT2ADRD3
SCHEMBL20765555 0.72 ALDH1A1 (0.66) ALDH1A1KDM4EHTTSMN1; SMN2USP2
SCHEMBL20765826 0.71 BCHE (0.41) ALDH1A1KDM4EROCK2POLB
SCHEMBL20765824 0.71 BCHE (0.41) ALDH1A1KDM4EROCK2POLB
SCHEMBL10007463 0.71 PKM (0.61) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed