SCHEMBL20765718

SCHEMBL20765718

Cc1nc2ccc(C(=O)N3CCN(C(=O)c4ccccc4)CC3)cc2[nH]1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.67
HPGD P15428 2/20 0.67
POLB P06746 1/20 0.67
RAB9A P51151 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
HSP90AA1 P07900 1/20 0.62
ESR2 Q92731 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
HSD11B1 P28845 2/20 0.53
ACACB O00763 4/20 0.53
ACACA Q13085 4/20 0.53
GHSR Q92847 1/20 0.52
BCHE P06276 2/20 0.52
ACHE P22303 2/20 0.52
MGLL Q99685 1/20 0.52
HTR2B P41595 1/20 0.51
MAPK1 P28482 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PDGFRB P09619 1/20 0.50
FGFR1 P11362 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17468532 0.88 HRH4 (0.62) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2
SCHEMBL16598920 0.87 MAOB (0.56) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2
SCHEMBL20765540 0.85 ENPP2 (0.57) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2
SCHEMBL20765644 0.83 KMT2A (0.60) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2
SCHEMBL20774926 0.81 ALDH1A1 (0.50) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2
SCHEMBL12909208 0.81 ALDH1A1 (1.00) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2
SCHEMBL13290560 0.78 KMT2A (0.47) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2
SCHEMBL8262960 0.78 MEN1 (0.60) ALDH1A1HPGDPOLBFGFR1KDR
SCHEMBL16598917 0.78 MAOB (0.56) ALDH1A1HPGDRAB9ASMN1; SMN2MAPT
Carbamic Acid SCHEMBL29258949 0.77 ALDH1A1 (0.92) ALDH1A1HPGDPOLBRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed