Stilbamidine

Stilbamidine

SCHEMBL20787646

N=C(N)c1ccc(/C=C/c2ccc(C(=N)N)cc2)cc1.O=S(=O)(O)CCO.O=S(=O)(O)CCO

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.78
KDM4E B2RXH2 2/20 0.78
MAPT P10636 2/20 0.78
RAD52 P43351 1/20 0.78
UBE2N P61088 1/20 0.78
NPSR1 Q6W5P4 1/20 0.78
ALDH1A1 P00352 3/20 0.61
PRMT1 Q99873 2/20 0.61
PRMT5 O14744 1/20 0.61
HPGD P15428 1/20 0.61
CYP2C19 P33261 1/20 0.61
HSD17B10 Q99714 1/20 0.61
LMNA P02545 2/20 0.61
RAB9A P51151 2/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
NPC1 O15118 1/20 0.61
ALOX15 P16050 1/20 0.61
BRCA1 P38398 1/20 0.61
HTT P42858 1/20 0.61
GMNN O75496 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Stilbamidine SCHEMBL3934275 1.00 POLB (0.78) POLBKDM4EMAPTRAD52UBE2N
Hydroxystilbamidine SCHEMBL554644 0.88 POLB (1.00) POLBKDM4EMAPTRAD52UBE2N
Hydroxystilbamidine SCHEMBL10621745 0.88 POLB (1.00) POLBKDM4EMAPTRAD52UBE2N
Hydroxystilbamidine SCHEMBL10621740 0.88 POLB (1.00) POLBKDM4EMAPTRAD52UBE2N
Benzamidine SCHEMBL27925636 0.81 POLB (0.61) POLBKDM4EMAPTRAD52UBE2N
Benzamidine SCHEMBL5522150 0.81 POLB (0.61) POLBKDM4EMAPTRAD52UBE2N
SCHEMBL5522149 0.81 POLB (0.74) POLBKDM4EMAPTRAD52UBE2N
Stilbamidine SCHEMBL208655 0.78 PRMT1 (1.00) ALDH1A1PRMT1PRMT5HPGDCYP2C19
Stilbamidine SCHEMBL889782 0.78 PRMT1 (1.00) ALDH1A1PRMT1PRMT5HPGDCYP2C19
Propamidine SCHEMBL293021 0.77 ALDH1A1 (0.92) POLBKDM4EMAPTALDH1A1PRMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376074-B1 METHOD FOR IMPROVED BIOACTIVATION OF MEDICATIONS DRITTE PATENTPORTFOLIO BETEILI (DE) 2019-03-13 EP disclosed