SCHEMBL20831743

SCHEMBL20831743

Cc1ccccc1CN1CCN(c2cn[nH]c(=O)c2Cl)CCC1=O

nearest known ligand 0.83

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPC5 Q9UL62 18/20 0.83
KCNH2 Q12809 1/20 0.61
TRPC4 Q9UBN4 1/20 0.61
ALDH1A1 P00352 1/20 0.57
POLB P06746 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20831413 0.91 TRPC5 (1.00) TRPC5KCNH2TRPC4ALDH1A1
SCHEMBL20831741 0.86 ALDH1A1 (0.74) TRPC5KCNH2TRPC4ALDH1A1POLB
SCHEMBL20831742 0.85 TRPC5 (0.84) TRPC5KCNH2TRPC4ALDH1A1POLB
SCHEMBL20831568 0.84 TRPC5 (0.88) TRPC5KCNH2TRPC4POLB
SCHEMBL20831566 0.82 TRPC5 (0.84) TRPC5KCNH2TRPC4ALDH1A1POLB
SCHEMBL20831375 0.81 TRPC5 (1.00) TRPC5KCNH2TRPC4ALDH1A1
SCHEMBL20818563 0.81 TRPC5 (1.00) TRPC5KCNH2TRPC4
SCHEMBL30476379 0.81 TRPC5 (1.00) TRPC5KCNH2TRPC4
SCHEMBL20818405 0.79 POLB (0.68) TRPC5KCNH2TRPC4ALDH1A1POLB
SCHEMBL20831207 0.79 TRPC5 (1.00) TRPC5KCNH2TRPC4ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GFB (ABC), LLC 2023-06-29 US disclosed
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GFB (ABC), LLC 2023-06-29 US disclosed
WO-2019055966-A2 PYRIDAZINONES AND METHODS OF USE THEREOF GOLDFINCH BIO, INC. (US) 2019-03-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF PDXK, ATP6V1B1, REN TRPC5 1439/4885KCNH2 915/4885TRPC4 2143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.