SCHEMBL20846293

SCHEMBL20846293

FC(F)(F)Oc1ccccc1-c1c[nH]c2ncccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.61
TGFBR1 P36897 4/20 0.50
IKBKE Q14164 3/20 0.49
TBK1 Q9UHD2 3/20 0.49
PDPK1 O15530 3/20 0.49
BRD4 O60885 1/20 0.47
CDC7 O00311 4/20 0.47
CDK2 P24941 3/20 0.47
MAP4K4 O95819 3/20 0.47
PIM1 P11309 3/20 0.47
PRKACA P17612 3/20 0.47
GSK3B P49841 3/20 0.47
HIPK2 Q9H2X6 3/20 0.47
IRAK4 Q9NWZ3 2/20 0.47
CLK4 Q9HAZ1 2/20 0.47
ROCK2 O75116 1/20 0.47
CCNB2 O95067 3/20 0.45
CDK1 P06493 3/20 0.45
CCNB1 P14635 3/20 0.45
CCNB3 Q8WWL7 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL857542 0.81 BRD4 (0.64) DYRK1ATGFBR1IKBKETBK1PDPK1
SCHEMBL10124933 0.81 AURKB (0.54) DYRK1ABRD4CDK2MAP4K4PRKACA
SCHEMBL20846156 0.80 CAMKK2 (0.48) DYRK1ACDK2MAP4K4HIPK2IRAK4
SCHEMBL857733 0.79 TGFBR1 (0.51) DYRK1ATGFBR1IKBKETBK1PDPK1
SCHEMBL20846121 0.78 CCNB2 (0.59) DYRK1ATGFBR1IKBKETBK1PDPK1
SCHEMBL5618155 0.78 TGFBR1 (0.71) DYRK1ATGFBR1IKBKETBK1PDPK1
SCHEMBL27704617 0.78 GPR84 (0.53) CDK2PIM1PRKACACCNB2CDK1
SCHEMBL858127 0.78 DYRK1A (0.61) DYRK1ATGFBR1IKBKEPDPK1BRD4
SCHEMBL20293419 0.76 DYRK1A (1.00) DYRK1AIKBKETBK1BRD4CDC7
SCHEMBL20846166 0.76 CAMKK2 (0.46) DYRK1ACDK2CDK9CCNT1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057660-A1 INDOLE AND AZAINDOLE COMPOUNDS WITH SUBSTITUTED 6-MEMBERED ARYL AND HETEROARYL RINGS AS AGROCHEMICAL FUNGICIDES BASF SE (DE) 2019-03-28 WO disclosed