SCHEMBL20853019

SCHEMBL20853019

COCc1cc2cc(F)c(F)cc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
LOXL2 Q9Y4K0 3/20 0.37
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
GPR84 Q9NQS5 1/20 0.34
KDM5A P29375 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
CACNA1H O95180 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
DRD3 P35462 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
EIF4A3 P38919 1/20 0.31
EHMT2 Q96KQ7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26422975 0.79 GPR84 (0.38) MAPTLOXL2ALDH1A1GPR84EIF4A3
SCHEMBL764523 0.75 LOXL2 (0.33) LOXL2
SCHEMBL24414591 0.75 RHEB (0.41) LOXL2GPR84EIF4A3NPC1RAB9A
SCHEMBL30991851 0.75 RHEB (0.41) LOXL2GPR84EIF4A3NPC1RAB9A
SCHEMBL26262596 0.74 NR3C1 (0.34) LOXL2GPR84EIF4A3
SCHEMBL12056086 0.74 ALDH1A1 (0.38) MAPTLOXL2ALDH1A1GPR84DRD4
SCHEMBL12334164 0.73 LOXL2 (0.64) MAPTLOXL2ALDH1A1GAAHPGD
SCHEMBL14081528 0.73 FLT3 (0.47) LOXL2GAAALOX15SMN1; SMN2MTNR1A
SCHEMBL2111019 0.72 LOXL2 (0.58) MAPTLOXL2ALDH1A1HPGDSMN1; SMN2
SCHEMBL14493641 0.71 LOXL2 (0.62) MAPTLOXL2ALDH1A1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3684767-B1 HETEROCYCLIC COMPOUNDS AS PAD INHIBITORS Jubilant Epipad LLC (US) 2024-04-24 EP disclosed
WO-2019058393-A1 HETEROCYCLIC COMPOUNDS AS PAD INHIBITORS JUBILANT BIOSYS LIMITED (IN) 2019-03-28 WO disclosed