SCHEMBL208620

SCHEMBL208620

Fc1ccc2[c]noc2c1

nearest known ligand 0.32

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL208122 0.75 AHR (0.32)
SCHEMBL8613814 0.71 KDM4E (0.40) MAOB
SCHEMBL207600 0.62 AHR (0.37)
SCHEMBL4306677 0.61
SCHEMBL3412034 0.60 CYP1A2 (0.38) MAOB
SCHEMBL207898 0.59 HDAC8 (0.30)
SCHEMBL325358 0.59 ALDH1A1 (0.41)
SCHEMBL5206649 0.59 PGR (0.38) MAOB
SCHEMBL978860 0.58 TP53 (0.32)
SCHEMBL208062 0.58 MAP2K4 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 168 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220048910-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES, INC. (US) 2022-02-17 US claimed
EP-3946345-A1 METHODS OF TREATING NEUROPATHIC PAIN Intra-Cellular Therapies, Inc. (US) 2022-02-09 EP claimed
CN-113905737-A Method of treating neuropathic pain 细胞内治疗公司 2022-01-07 CN claimed
EP-3914235-A2 METHODS OF TREATING ADDICTION Intra-Cellular Therapies, Inc. (US) 2021-12-01 EP claimed
EP-3897621-A1 ORGANIC COMPOUNDS Intra-Cellular Therapies, Inc. (US) 2021-10-27 EP claimed
CN-113329742-A Method for treating addiction 细胞内治疗公司 2021-08-31 CN claimed
WO-2020206391-A1 METHODS OF TREATING NEUROPATHIC PAIN INTRA-CELLULAR THERAPIES, INC. (US) 2020-10-08 WO claimed
WO-2020154519-A2 METHODS OF TREATING ADDICTION INTRA-CELLULAR THERAPIES, INC. (US) 2020-07-30 WO claimed
WO-2020132605-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES, INC. (US) 2020-06-25 WO claimed
US-9238658-B2 Substituted piperidinyl-carboxamide derivatives useful as SCD 1 inhibitors JANSSEN PHARMACEUTICA NV (BE) 2016-01-19 US claimed
EP-1776349-A2 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE) JANSSEN PHARMACEUTICA N.V. (BE) 2007-04-25 EP claimed
US-20060079687-A1 Novel 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (BACE) JANSSEN PHARMACEUTICA, N.V. (BE) 2006-04-13 US claimed
WO-2006017836-A2 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE) JANSSEN PHARMACEUTICA, N.V. (BE) 2006-02-16 WO claimed
EP-0700396-A1 PIPERIDINE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1996-03-13 EP claimed
US-5478845-A Inhibit dopamine or 5-hydroxytryptamine receptor binding NOVO NORDISK A/S (DK) 1995-12-26 US claimed
WO-1994027996-A1 1,2,5-THIADIAZOLE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1994-12-08 WO claimed
WO-1994027992-A1 PIPERIDINE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1994-12-08 WO claimed
WO-1994027994-A1 PIPERIDINE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1994-12-08 WO claimed
EP-0377528-B1 Piperidines, process for their preparation and pharmaceutical compounds containing them LIPHA (FR) 1993-12-08 EP claimed
US-5001134-A Piperidines, processes of preparation and medications containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1991-03-19 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060079687-A1 Novel 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (BACE) BACE2, BACE1, APP MAOB 532/4885
US-20220048910-A1 ORGANIC COMPOUNDS OPRD1, OPRM1, HTR2C MAOB 130/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.