SCHEMBL20870495

SCHEMBL20870495

CCCC(O)CCc1cc(CC)ccc1NC

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
HTR1A P08908 1/20 0.34
TRPA1 O75762 1/20 0.33
AKT1 P31749 1/20 0.32
STAT3 P40763 1/20 0.31
GAA P10253 1/20 0.31
BACE1 P56817 1/20 0.30
HPGD P15428 1/20 0.30
METAP2 P50579 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22061268 0.90 METAP2 (0.33) TRPA1AKT1STAT3GAABACE1
SCHEMBL22061292 0.90 METAP2 (0.33) TRPA1AKT1STAT3GAABACE1
SCHEMBL20006392 0.81 TRPA1 (0.36) HTR1ATRPA1AKT1BACE1METAP2
SCHEMBL20870189 0.80 PDK2 (0.33) TRPA1AKT1GAAMETAP2
SCHEMBL20870405 0.79 KCNH2 (0.36) TRPA1AKT1
SCHEMBL22279702 0.79 SKP2 (0.36) TAS1R3TAS1R1HTR1ATRPA1AKT1
SCHEMBL9449596 0.75 TRPA1 (0.40) TRPA1AKT1GAABACE1METAP2
SCHEMBL21228550 0.73 LMNA (0.39) GAAMETAP2
SCHEMBL20870143 0.73 AR (0.36) TRPA1AKT1BACE1METAP2
SCHEMBL22279892 0.71 HTR1A (0.42) HTR1ATRPA1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019063015-A1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUND WHICH ACTS AS RORγ INHIBITOR 正大天晴药业集团股份有限公司 2019-04-04 WO disclosed