SCHEMBL20880758

SCHEMBL20880758

Nc1cccc2c1OCCNC2=O

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.54
FABP6 P51161 1/20 0.43
PARP10 Q53GL7 4/20 0.40
PARP11 Q9NR21 4/20 0.40
PDPK1 O15530 1/20 0.40
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
CDK5 Q00535 2/20 0.38
DYRK1A Q13627 2/20 0.38
CLK4 Q9HAZ1 2/20 0.38
PIM1 P11309 1/20 0.38
CSNK1A1 P48729 1/20 0.38
ROCK1 Q13464 1/20 0.38
LRRK2 Q5S007 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
LTK P29376 1/20 0.33
MST1R Q04912 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21333792 0.80 FABP6 (0.50) PARP1FABP6PARP10PARP11PDPK1
SCHEMBL21999476 0.80 PARP1 (0.54) PARP1FABP6PARP10PARP11PDPK1
SCHEMBL2985573 0.80 PARP1 (0.54) PARP1FABP6PARP10PARP11PDPK1
SCHEMBL2983974 0.76 ALPL (0.46) PARP1FABP6PARP10PARP11
SCHEMBL1027825 0.75 DRD2 (0.39) PARP1
SCHEMBL21461173 0.75 S100A4 (0.42) PARP1FABP6PARP10PARP11PDPK1
SCHEMBL2085452 0.75 PARP1 (0.44) PARP1FABP6PARP10PARP11PDPK1
SCHEMBL2060616 0.74 FABP6 (0.55) PARP1FABP6PARP10PARP11
SCHEMBL3993011 0.74 LMNA (0.44) PARP1
SCHEMBL12714478 0.73 FABP6 (0.43) PARP1FABP6CDK5CLK4CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227263-B1 CXCR7 RECEPTOR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2019-04-10 EP disclosed