SCHEMBL20904792

SCHEMBL20904792

O=C(CC(=O)C(F)(F)F)c1nncs1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 3/20 0.45
PLOD3 O60568 2/20 0.45
PLOD1 Q02809 2/20 0.45
CES1 P23141 2/20 0.42
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP1A2 P05177 2/20 0.32
TSHR P16473 1/20 0.32
POLB P06746 4/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
ESR2 Q92731 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321698 0.72 PLOD2 (0.49) PLOD2PLOD3PLOD1CES1ALDH1A1
SCHEMBL17951545 0.68 CES1 (0.42) CES1ALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL23511768 0.66
SCHEMBL1279224 0.65
SCHEMBL6979211 0.64 RAB9A (0.58) ALDH1A1HPGDTSHRPOLBSMN1; SMN2
SCHEMBL195358 0.63 ERCC5 (0.59) PLOD2PLOD3PLOD1CES1ALDH1A1
SCHEMBL18622294 0.63 PLOD2 (0.55) PLOD2PLOD3PLOD1CES1KDM4E
SCHEMBL751818 0.62 GSK3B (0.56) PLOD2PLOD3PLOD1CES1ALDH1A1
SCHEMBL10631235 0.62 ERCC5 (0.57) PLOD2PLOD3PLOD1CES1ALDH1A1
SCHEMBL21408730 0.62 PLOD2 (0.67) PLOD2PLOD3PLOD1CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10835895-B2 Compound and synthesis method therefor THE UNIVERSITY OF TOKYO (JP) 2020-11-17 US disclosed
US-20190111418-A1 COMPOUND AND SYNTHESIS METHOD THEREFOR THE UNIVERSITY OF TOKYO (JP) 2019-04-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10835895-B2 Compound and synthesis method therefor GOT1, GOT2, SLC39A11 PLOD2 3759/4885PLOD3 4837/4885PLOD1 3345/4885
US-20190111418-A1 COMPOUND AND SYNTHESIS METHOD THEREFOR GOT1, GOT2, SLC39A11 PLOD2 3851/4885PLOD3 4841/4885PLOD1 3481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.