SCHEMBL209090

SCHEMBL209090

CC(C)[Si](OC1CCC([C@@H](c2ccc(-c3ccc(C(=O)O)c(Cl)c3)cc2Cl)C2CCNC2=O)CC1)(C(C)C)C(C)C

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.33
PRKAB2 O43741 2/20 0.32
PRKAG1 P54619 2/20 0.32
PRKAA2 P54646 2/20 0.32
PRKAA1 Q13131 2/20 0.32
PRKAG3 Q9UGI9 2/20 0.32
PRKAG2 Q9UGJ0 2/20 0.32
PRKAB1 Q9Y478 2/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
AKR1C2 P52895 1/20 0.31
AKR1C1 Q04828 1/20 0.31
MEN1 O00255 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL208541 0.82 SRD5A2 (0.32) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4060990 0.82 SRD5A2 (0.32) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4191602 0.81 XDH (0.35) XDHPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL207570 0.78 MAP2K4 (0.35)
SCHEMBL1092228 0.77 PDE4A (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL1094081 0.77 PDE4A (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL2993023 0.73 PDE4D (0.37) ADRB1ADRB3
SCHEMBL208946 0.73 P2RX7 (0.38) MEN1KMT2A
SCHEMBL1093033 0.72 PSD (0.34)
SCHEMBL3544149 0.72 KDM4E (0.37) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088776-B2 Biphenyl amide lactam derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1 ELI LILLY AND COMPANY (US) 2012-01-03 US disclosed
US-20090156571-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156571-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 HSD11B1, HSD17B1, HSD11B2 XDH 950/4885PRKAB2 1822/4885PRKAG1 813/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.