SCHEMBL20914549

SCHEMBL20914549

O=C(O)c1ccccc1-c1cc(Cn2cccn2)cc(-c2ccccc2C(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.54
UCHL5 Q9Y5K5 5/20 0.50
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
AGTR1 P30556 1/20 0.45
AGTR2 P50052 1/20 0.45
MEN1 O00255 1/20 0.44
TSHR P16473 1/20 0.44
KMT2A Q03164 1/20 0.44
GRK6 P43250 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
PPARG P37231 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20914488 0.76 UCHL5 (0.50) UCHL5AGTR1AGTR2MEN1KMT2A
SCHEMBL30284989 0.76 MEN1 (0.53) HTTHDAC1HDAC6AGTR1AGTR2
SCHEMBL20914481 0.76 MEN1 (0.53) HTTHDAC1HDAC6AGTR1AGTR2
SCHEMBL15155447 0.76 HTT (0.56) HTTHDAC1HDAC6MEN1TSHR
SCHEMBL30047867 0.74 ALDH1A1 (0.59) MEN1TSHRKMT2ACA12CA1
SCHEMBL139845 0.74 ALDH1A1 (0.59) MEN1TSHRKMT2ACA12CA1
SCHEMBL7081878 0.74 HTT (0.75) HTTHDAC1HDAC6MEN1TSHR
SCHEMBL20914432 0.72 BRS3 (0.45) AGTR1AGTR2
SCHEMBL297475 0.72 FOLH1 (0.49) UCHL5
SCHEMBL3584847 0.71 HDAC1 (0.70) HTTHDAC1HDAC6MEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10696635-B2 Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates THE SCRIPPS RESEARCH INSTITUTE (US) 2020-06-30 US disclosed
US-20190119212-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS THE SCRIPPS RESEARCH INSTITUTE 2019-04-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190119212-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS AHR, PAH, DOHH HTT 504/4885UCHL5 781/4885HDAC1 1011/4885
US-10696635-B2 Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates PAH, AHR, DDC HTT 686/4885UCHL5 1032/4885HDAC1 1111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.