SCHEMBL20914488

SCHEMBL20914488

O=C(O)c1ccccc1-c1cc(Cn2cc3ccccc3n2)cc(-c2ccccc2C(=O)O)c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
UCHL5 Q9Y5K5 5/20 0.50
PARP1 P09874 1/20 0.45
PPARG P37231 4/20 0.43
AGTR1 P30556 2/20 0.41
AGTR2 P50052 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20937661 0.86 SLC6A3 (0.49) UCHL5PARP1AGTR1AGTR2KDM4E
SCHEMBL30285127 0.86 SLC6A3 (0.49) UCHL5PARP1AGTR1AGTR2KDM4E
SCHEMBL30285026 0.78 SLC6A3 (0.50) PARP1AGTR1AGTR2KMT2A
SCHEMBL19475034 0.78 SLC6A3 (0.50) PARP1AGTR1AGTR2KMT2A
SCHEMBL20914549 0.76 HTT (0.54) UCHL5PPARGAGTR1AGTR2MEN1
SCHEMBL19512905 0.76 UCHL5 (0.42) UCHL5PARP1AGTR1AGTR2
SCHEMBL19475067 0.73 PARP1 (0.51) PARP1MEN1KMT2A
SCHEMBL15774394 0.73 PTPN1 (0.48) PARP1NPC1RAB9ASMN1; SMN2
SCHEMBL139845 0.72 ALDH1A1 (0.59) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL30047867 0.72 ALDH1A1 (0.59) KDM4EALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10696635-B2 Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates THE SCRIPPS RESEARCH INSTITUTE (US) 2020-06-30 US disclosed
US-20190119212-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS THE SCRIPPS RESEARCH INSTITUTE 2019-04-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190119212-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS AHR, PAH, DOHH UCHL5 781/4885PARP1 2042/4885PPARG 98/4885
US-10696635-B2 Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates PAH, AHR, DDC UCHL5 1032/4885PARP1 2563/4885PPARG 200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.