SCHEMBL20928443

SCHEMBL20928443

Cc1cccc(-c2cccc(C3Cc4ccc(Br)cc4O3)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 3/20 0.40
MAOB P27338 8/20 0.39
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 1/20 0.37
SLC5A2 P31639 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
RECQL P46063 1/20 0.36
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.34
FYN P06241 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
ALOX15B O15296 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
BACE1 P56817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20928108 0.81 FFAR1 (0.49) FFAR1RAB9AKMT2A
SCHEMBL20928517 0.81 MAPK1 (0.36) MAOBMAPK1ALDH1A1SLC5A2TP53
SCHEMBL23320409 0.78 LMNA (0.56) MAOBALDH1A1CYP3A4MAPTRAB9A
SCHEMBL28922327 0.78 LMNA (0.56) MAOBALDH1A1CYP3A4MAPTRAB9A
SCHEMBL20928142 0.76 FFAR1 (0.42) FFAR1MAOBALDH1A1MAPT
SCHEMBL14862016 0.75 MAOB (0.52) MAOBALDH1A1RAB9AKMT2ANPC1
SCHEMBL31346101 0.70 FFAR1 (0.38) FFAR1MAOB
SCHEMBL29165038 0.70 LMNA (0.50) MAOBALDH1A1TP53MAPTRAB9A
SCHEMBL31346096 0.70 FFAR1 (0.40) FFAR1MAOBALDH1A1MAPTKMT2A
SCHEMBL31345958 0.69 KDM1A (0.38) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019076343-A1 PD-1/PD-L1 SMALL-MOLECULE INHIBITOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海长森药业有限公司 2019-04-25 WO disclosed