SCHEMBL20931111

SCHEMBL20931111

C/C=C\c1cccc(C(C)Br)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.37
CYP3A4 P08684 3/20 0.34
ATM Q13315 2/20 0.34
NFE2L2 Q16236 3/20 0.33
TYR P14679 2/20 0.33
HPGD P15428 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 4/20 0.32
KDM4E B2RXH2 2/20 0.32
TP53 P04637 2/20 0.32
MAPT P10636 2/20 0.32
HTT P42858 2/20 0.32
MDM4 O15151 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
ALOX15 P16050 1/20 0.32
ALOX12 P18054 1/20 0.32
CA5A P35218 1/20 0.32
HDAC4 P56524 1/20 0.32
MDM2 Q00987 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14051358 0.84 TYR (0.46) CNR2CYP3A4ATMNFE2L2TYR
SCHEMBL8769118 0.78 TP53 (0.50) ALDH1A1TP53HDAC8TDP1TSHR
SCHEMBL29756201 0.78 ALDH1A1 (0.50) TYRSMN1; SMN2ALDH1A1CA1CA2
SCHEMBL7935947 0.78 CNR2 (0.42) CNR2CYP3A4ATMNFE2L2TYR
SCHEMBL11518269 0.78 HDAC4 (0.51) CNR2CYP3A4ATMTYRHPGD
SCHEMBL10447240 0.77 TAAR1 (0.50) CNR2ATMHPGDSMN1; SMN2HDAC4
SCHEMBL8897527 0.76 HDAC4 (0.37) CYP3A4TYRHPGDSMN1; SMN2ALDH1A1
SCHEMBL335942 0.76 CNR2 (0.50) CNR2CYP3A4ATMNFE2L2TYR
SCHEMBL29033283 0.76 CNR2 (0.50) CNR2CYP3A4ATMNFE2L2TYR
SCHEMBL335941 0.76 CNR2 (0.50) CNR2CYP3A4ATMNFE2L2TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019079578-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USES AMGEN INC. (US) 2019-04-25 WO disclosed