SCHEMBL2094079

SCHEMBL2094079

O=CNc1c(Cl)cccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
GAA P10253 4/20 0.39
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2A6 P11509 1/20 0.38
TYK2 P29597 1/20 0.37
P2RX7 Q99572 1/20 0.37
LMNA P02545 2/20 0.36
TSHR P16473 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2C P18825 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13623166 0.87 ALDH1A1 (0.46) ALDH1A1MEN1KMT2ATDP1CYP2A6
SCHEMBL7528740 0.85 GAA (0.46) ALDH1A1MEN1KMT2ATDP1GAA
SCHEMBL16240433 0.85 TDP1 (0.40) ALDH1A1MEN1KMT2ATDP1GAA
SCHEMBL27851425 0.85 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ATDP1GAA
SCHEMBL21461560 0.85 GAA (0.45) ALDH1A1MEN1KMT2ATDP1GAA
SCHEMBL11614677 0.80 PTGS2 (0.46) ALDH1A1MEN1KMT2ATDP1TYK2
SCHEMBL2097678 0.75 ERN1 (0.40) ALDH1A1MEN1KMT2ATDP1GAA
SCHEMBL11915484 0.75 CYP1A2 (0.38) ALDH1A1MEN1KMT2ATDP1GAA
SCHEMBL448938 0.75 MEN1 (0.50) ALDH1A1MEN1KMT2ATDP1MAPT
SCHEMBL20341641 0.73 TDP1 (0.38) ALDH1A1MEN1KMT2ATDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
US-4935515-A ANTIARRHYTHMIA AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1990-06-19 US claimed
EP-0358749-A1 1,4-SUBSTITUTED-2,3,5,6-TETRAHYDRO 1,3,6]TRIAZOCINO 1,2-a]BENZIMIDAZOLES AND INTERMEDIATES THEREFOR AMERICAN HOME PRODUCTS CORPORATION (US) 1990-03-21 EP claimed
WO-1989008111-A1 1,4-SUBSTITUTED-2,3,5,6-TETRAHYDRO[1,3,6]TRIAZOCINO[1,2-a]BENZIMIDAZOLES AND INTERMEDIATES THEREFOR AMERICAN HOME PRODUCTS CORPORATION (US) 1989-09-08 WO claimed
US-4801706-A ANTIARRHYTHMIA HYPOTENSIVE AMERICAN HOME PRODUCTS CORPORATION (US) 1989-01-31 US claimed
JP-55072152-A None JP disclosed
US-20260007638-A1 STABLE PHARMACEUTICAL COMPOSITIONS OF CLONIDINE AZURITY PHARMACEUTICALS, INC. (US) 2026-01-08 US disclosed
US-12440474-B2 Stable pharmaceutical compositions of clonidine AZURITY PHARMACEUTICALS, INC. (US) 2025-10-14 US disclosed
US-20250152558-A1 STABLE PHARMACEUTICAL COMPOSITIONS OF CLONIDINE SLAYBACK PHARMA LLC (US) 2025-05-15 US disclosed
US-12233049-B2 Stable pharmaceutical compositions of clonidine SLAYBACK PHARMA LLC (US) 2025-02-25 US disclosed
US-20230149359-A1 STABLE PHARMACEUTICAL COMPOSITIONS OF CLONIDINE AZURITY PHARMACEUTICALS, INC. 2023-05-18 US disclosed
US-20230149359-A1 STABLE PHARMACEUTICAL COMPOSITIONS OF CLONIDINE AZURITY PHARMACEUTICALS, INC. 2023-05-18 US disclosed
EP-0002010-B1 DERIVATIVES OF 2-IMINO-IMIDAZOLIDINE, PROCESSES FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND INTERMEDIATES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-07-14 EP disclosed
EP-0003259-B1 N-FORMYLANILIDO AROMATIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PROCESS FOR THE PREPARATION OF THE CORRESPONDING N-PHENYL AROMATIC AMINO COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-03-24 EP disclosed
US-4292446-A N-FORMYLANILINO AROMATICS, DIPHENYLAMINE INTERMEDIATES, PESTICIDES, PREPARATION FROM FORMANILIDES AND HALOAROMATICS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1981-09-29 US disclosed
US-4244957-A HYPOTENSIVE AGENTS HOFFMAN-LA ROCHE INC. (US) 1981-01-13 US disclosed
JP-S5572152-A PREPARATION OF 2-(2,6-DICHLOROANILINO)PHENYLACETIC ACID AND ITS SALT TAIYO YAKUHIN KOGYO KK 1980-05-30 JP disclosed
EP-0003259-A1 N-Formylanilido aromatic compounds, process for their preparation and process for the preparation of the corresponding N-phenyl aromatic amino compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-08 EP disclosed
EP-0002010-A1 Derivatives of 2-imino-imidazolidine, processes for their preparation, pharmaceutical compositions containing them and intermediates F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-05-30 EP disclosed
US-4024259-A 3-Anilino-2,4-diazabicyclo[3.2.1]octenes AMERICAN HOECHST CORPORATION (US) 1977-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12440474-B2 Stable pharmaceutical compositions of clonidine ADRA2C, SLC6A2, ADRA2A ALDH1A1 1934/4885MEN1 2539/4885KMT2A 2550/4885
US-12233049-B2 Stable pharmaceutical compositions of clonidine ADRA2C, SLC6A2, ADRA2A ALDH1A1 1934/4885MEN1 2539/4885KMT2A 2550/4885
US-20260007638-A1 STABLE PHARMACEUTICAL COMPOSITIONS OF CLONIDINE CHRM2, GLP1R, CHRM1 ALDH1A1 2274/4885MEN1 948/4885KMT2A 590/4885
US-20250152558-A1 STABLE PHARMACEUTICAL COMPOSITIONS OF CLONIDINE ADRA2C, SLC6A2, ADRA2A ALDH1A1 1934/4885MEN1 2539/4885KMT2A 2550/4885
US-20230149359-A1 STABLE PHARMACEUTICAL COMPOSITIONS OF CLONIDINE ADRA2C, SLC6A2, ADRA2A ALDH1A1 1973/4885MEN1 2477/4885KMT2A 2500/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.