Tabimorelin

Tabimorelin

SCHEMBL209441

CNC(=O)[C@@H](Cc1ccccc1)N(C)C(=O)[C@@H](Cc1ccc2ccccc2c1)N(C)C(=O)/C=C/CC(C)(C)N

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CYP3A4GHSR

The experimentally established mechanism targets of Tabimorelin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GHSR known ✓ Q92847 8/20 0.65
FCER2 P06734 3/20 0.41
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tabimorelin SCHEMBL29440097 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
SCHEMBL6316837 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
Tabimorelin SCHEMBL29899698 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
Tabimorelin SCHEMBL209442 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
Tabimorelin SCHEMBL13575741 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
SCHEMBL6316843 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
Tabimorelin SCHEMBL7982376 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
Tabimorelin SCHEMBL4435323 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
Tabimorelin SCHEMBL22345096 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8
Tabimorelin SCHEMBL29958795 1.00 GHSR (0.65) GHSRFCER2MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 553 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12629363-B2 Prophylaxis and treatment of angioedema PHARVARIS GMBH (CH) 2026-05-19 US claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
EP-4604743-A1 FORMULATED FOOD PRODUCTS VitaKey Inc. (US) 2025-08-27 EP claimed
US-20240325404-A1 TREATMENT OF INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2024-10-03 US claimed
WO-2024086307-A1 FORMULATED FOOD PRODUCTS VITAKEY INC. (US) 2024-04-25 WO claimed
WO-2024086306-A1 FORMULATED FOOD PRODUCTS VITAKEY INC. (US) 2024-04-25 WO claimed
US-20230330187-A1 USE OF GHRELIN OR GHRELIN VARIANT FOR INCREASING DOSE INTENSITY OF CHEMOTHERAPEUTIC AGENTS IN PATIENTS WITH CANCER OXEIA BIOPHARMACEUTICALS INC (US) 2023-10-19 US claimed
WO-2023161326-A1 COMPOUND FOR USE IN AND METHODS OF TREATMENT OF INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2023-08-31 WO claimed
US-20220370471-A1 COMPOSITION AND METHOD FOR TREATMENT OF HIPPOCAMPAL SYNAPSE DYSFUNCTION AND COGNITIVE DEFICITS IN ALZHEIMER'S DISEASE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-11-24 US claimed
WO-2022226116-A1 GHRELIN TREATMENT OF BRAIN DYSFUNCTION DUE TO VIRAL INFECTION OXEIA BIOPHARMACEUTICALS, INC. (US) 2022-10-27 WO claimed
JP-2002521322-A 2002-07-16 JP claimed
US-20020022649-A1 STABLE PHARMACEUTICAL FORMULATION HELSINN THERAPEUTICS (U.S.), INC. 2002-02-21 US claimed
US-6281247-B1 GLANDULAR DISORDERS; ANIMAL GROWTH REGULATORS NOVO NORDISK A/S (DK) 2001-08-28 US claimed
EP-1098636-A1 A WET GRANULATION METHOD FOR PREPARING A STABLE PHARMACEUTICAL FORMULATION NOVO NORDISK A/S (DK) 2001-05-16 EP claimed
EP-1060190-A1 NEW SALT FORMS OF (2E)- 5-AMINO-5- METHYLHEX-2- ENOIC ACID N-METHYL-N-((1R)-1-(N- METHYL-N-((1R)-1-(METHYLCARBAMOYL)-2- PHENYLETHYL)CARBAMOYL)-2- (2-NAPHTYL)ETHYL)AMIDE NOVO NORDISK A/S (DK) 2000-12-20 EP claimed
WO-2000004880-A1 A WET GRANULATION METHOD FOR PREPARING A STABLE PHARMACEUTICAL FORMULATION NOVO NORDISK A/S (DK) 2000-02-03 WO claimed
US-5977178-A Compounds with growth hormone releasing properties NOVO NORDISK A/S (DK) 1999-11-02 US claimed
WO-1999045029-A1 NEW SALT FORMS OF (2E)- 5-AMINO-5- METHYLHEX-2- ENOIC ACID N-METHYL-N-((1R)-1-(N- METHYL-N-((1R)-1-(METHYLCARBAMOYL)-2- PHENYLETHYL)CARBAMOYL)-2- (2-NAPHTYL)ETHYL)AMIDE NOVO NORDISK A/S (DK) 1999-09-10 WO claimed
EP-0869974-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1998-10-14 EP claimed
WO-1997023508-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1997-07-03 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240325404-A1 TREATMENT OF INFLAMMATORY DISEASES IFNAR1, IFNG, IRF3 GHSR 1226/4885FCER2 217/4885MMP9 1494/4885
US-20020022649-A1 STABLE PHARMACEUTICAL FORMULATION GRN, COG6, UGGT1 GHSR 617/4885FCER2 2372/4885MMP9 3352/4885
US-12629363-B2 Prophylaxis and treatment of angioedema BDKRB2, BDKRB1, HRH2 GHSR 639/4885FCER2 30/4885MMP9 1143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.