SCHEMBL21032545

SCHEMBL21032545

CCn1c(C)c(-c2csc3ccc(F)cc23)c2cc(C)ccc21

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.39
TP53 P04637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTGDR2 Q9Y5Y4 12/20 0.36
CYP2C9 P11712 2/20 0.36
PTGDR Q13258 1/20 0.36
PMM2 O15305 1/20 0.34
G6PD P11413 1/20 0.34
MPI P34949 1/20 0.34
PHOSPHO1 Q8TCT1 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
PTGS1 P23219 2/20 0.34
SLC6A4 P31645 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21032411 0.88 HTR6 (0.46) MAPTKDM4EMAPK1L3MBTL1PTGDR2
SCHEMBL21031946 0.85 PTGDR2 (0.53) PTGDR2CYP2C9PTGDRPTGS1SLC6A4
SCHEMBL24179951 0.80 PTGDR2 (0.56) PTGDR2CYP2C9PTGDR
SCHEMBL21032472 0.80 PTGDR2 (0.48) MAPTTP53PTGDR2PTGS1
SCHEMBL21032707 0.78 MAPK14 (0.43) MAPTKDM4EMAPK1L3MBTL1PTGDR2
SCHEMBL21032706 0.76 PTGDR2 (0.36) MAPTKDM4EMAPK1L3MBTL1PTGDR2
SCHEMBL20631884 0.76 KDM4E (0.50) MAPTKDM4EMAPK1L3MBTL1ALDH1A1
SCHEMBL21032166 0.75 PTGDR2 (0.59) PTGDR2CYP2C9PTGDRPTGS1
SCHEMBL21032557 0.74 PTGDR2 (0.54) PTGDR2CYP2C9PTGDR
SCHEMBL24180036 0.73 PTGDR2 (0.63) PTGDR2CYP2C9PTGS1SLC6A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed