SCHEMBL21035631

SCHEMBL21035631

COC(=O)[C@@H]1CN([C@H](C)c2ccc(-c3ccc(Cl)cc3)cc2)CCN1S(=O)(=O)c1ccc(OCC2CCCCC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.42
KCNQ1 P51787 2/20 0.42
CHRM1 P11229 2/20 0.42
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
BCL2L1 Q07817 1/20 0.41
MCL1 Q07820 1/20 0.41
MMP3 P08254 3/20 0.40
MMP1 P03956 3/20 0.40
MMP7 P09237 2/20 0.40
MMP13 P45452 2/20 0.40
MEN1 O00255 1/20 0.40
ADAM17 P78536 1/20 0.40
RGS12 O14924 1/20 0.40
MMP9 P14780 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21035630 1.00 CHRM2 (0.42) CHRM2KCNQ1CHRM1KMT2AALDH1A1
SCHEMBL21035632 0.92 CHRM2 (0.43) CHRM2KCNQ1CHRM1KMT2AALDH1A1
SCHEMBL21035634 0.92 CHRM2 (0.43) CHRM2KCNQ1CHRM1KMT2AALDH1A1
SCHEMBL21002001 0.87 GHSR (0.45) CHRM2KCNQ1CHRM1KMT2ANPSR1
SCHEMBL21035633 0.87 GHSR (0.45) CHRM2KCNQ1CHRM1KMT2ANPSR1
SCHEMBL21001945 0.87 GHSR (0.45) CHRM2KCNQ1CHRM1KMT2ANPSR1
SCHEMBL21035573 0.82 LMNA (0.48) KMT2AALDH1A1NPSR1MMP3MMP1
SCHEMBL21035356 0.82 LMNA (0.48) KMT2AALDH1A1NPSR1MMP3MMP1
SCHEMBL21035083 0.81 MMP1 (0.46) KCNQ1KMT2ANPSR1BCL2L1MCL1
SCHEMBL21035659 0.81 MMP1 (0.46) KCNQ1KMT2ANPSR1BCL2L1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed