SCHEMBL21048757

SCHEMBL21048757

COc1ccc(N(S(=O)(=O)c2ccccc2)S(=O)(=O)c2ccccc2)c(C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 5/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
PGR P06401 3/20 0.43
TAS2R14 Q9NYV8 3/20 0.43
NFE2L2 Q16236 4/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 1/20 0.41
STAT3 P40763 1/20 0.41
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21048771 0.81 GLA (0.41) PGRL3MBTL1KDM4EMAPK1POLB
SCHEMBL31267493 0.79 MAPT (0.55) PGRTSHRPOLBMAPT
SCHEMBL21048811 0.78 CYP3A4 (0.47) KEAP1CYP3A4CYP2C9CYP2C19TAS2R14
SCHEMBL17259042 0.72 PGR (0.57) KEAP1PGRTAS2R14NFE2L2L3MBTL1
SCHEMBL7829381 0.71 MAPT (0.52) KEAP1PGRTAS2R14NFE2L2TSHR
SCHEMBL19848182 0.69 KEAP1 (0.47) KEAP1CYP3A4CYP2C9CYP2C19PGR
SCHEMBL21734440 0.69 KEAP1 (0.59) KEAP1CYP2C9PGRTAS2R14NFE2L2
SCHEMBL19416820 0.68 ALDH1A1 (0.60) KEAP1PGRL3MBTL1KDM4EPOLB
SCHEMBL7534915 0.68 KDM4E (0.52) KDM4EGAAMAPT
SCHEMBL28802576 0.67 MAOA (0.49) CYP3A4CYP2C9CYP2C19PGRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed