SCHEMBL21048811

SCHEMBL21048811

N#Cc1ccccc1N(S(=O)(=O)c1ccccc1)S(=O)(=O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 4/20 0.46
HTT P42858 1/20 0.46
APOBEC3G Q9HC16 1/20 0.42
TAS2R14 Q9NYV8 1/20 0.40
KDM4E B2RXH2 1/20 0.39
RORC P51449 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
HTR6 P50406 2/20 0.36
C5AR1 P21730 1/20 0.36
TSHR P16473 1/20 0.35
MCL1 Q07820 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2892311 0.83 C5AR1 (0.53) ALDH1A1HTTKDM4EKEAP1LMNA
SCHEMBL17258696 0.78 ALDH1A1 (0.49) ALDH1A1HTTKDM4ERORCLMNA
SCHEMBL21048757 0.78 KEAP1 (0.45) CYP3A4CYP2C9CYP2C19TAS2R14KDM4E
SCHEMBL21048806 0.75 ALDH1A1 (0.46) ALDH1A1HTTKDM4ERORCHPGD
SCHEMBL5853978 0.72 TEAD1 (0.49) CYP3A4CYP2C9CYP2C19ALDH1A1APOBEC3G
SCHEMBL5853971 0.72 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19ALDH1A1APOBEC3G
SCHEMBL16550141 0.72 APOBEC3G (0.52) CYP3A4CYP2C9CYP2C19ALDH1A1APOBEC3G
SCHEMBL16539764 0.70 ALDH1A1 (0.41) CYP3A4CYP2C9CYP2C19ALDH1A1HTT
SCHEMBL29827525 0.69 TSHR (0.48) CYP3A4CYP2C9CYP2C19ALDH1A1HTT
SCHEMBL8974476 0.69 ALDH1A1 (0.46) CYP3A4CYP2C9CYP2C19ALDH1A1APOBEC3G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed