SCHEMBL21078258

SCHEMBL21078258

CCCC(CCC)C(=O)N1CCN(C)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.46
TDP1 Q9NUW8 3/20 0.45
CYP1A2 P05177 1/20 0.45
HSD17B10 Q99714 1/20 0.42
CYP2C19 P33261 1/20 0.42
CHRM1 P11229 4/20 0.41
AKR1A1 P14550 1/20 0.41
CHRM3 P20309 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
ADRA1A P35348 1/20 0.41
HRH1 P35367 1/20 0.41
DRD3 P35462 1/20 0.41
SLC6A3 Q01959 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
KDM4E B2RXH2 3/20 0.41
CYP3A4 P08684 2/20 0.40
TSHR P16473 2/20 0.40
NFKB1 P19838 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26308166 0.93 ALDH1A1 (0.46) HTR1ATDP1CYP1A2HSD17B10CYP2C19
SCHEMBL20416320 0.92 CYP2C19 (0.47) HTR1ATDP1CYP1A2HSD17B10CYP2C19
SCHEMBL18782931 0.85 CA2 (0.44) HTR1ATDP1CYP1A2HSD17B10CYP2C19
SCHEMBL18949009 0.85 CA2 (0.44) HTR1ATDP1CYP1A2HSD17B10CYP2C19
SCHEMBL22628668 0.85 CA2 (0.44) HTR1ATDP1CYP1A2HSD17B10CYP2C19
SCHEMBL20444070 0.84 CA2 (0.47) HTR1ATDP1CYP1A2KDM4ETSHR
SCHEMBL4548032 0.83 CYP2C19 (0.57) HTR1ATDP1CYP1A2HSD17B10CYP2C19
SCHEMBL7503597 0.83 SLC6A3 (0.44) TDP1CYP2C19CHRM1AKR1A1CHRM3
SCHEMBL21428423 0.82 HSD17B10 (0.53) HTR1ATDP1CYP1A2HSD17B10CYP2C19
SCHEMBL6950102 0.82 HTR1A (0.44) HTR1ATDP1CYP1A2HSD17B10CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed