SCHEMBL21079230

SCHEMBL21079230

Brc1cccc2c1C[C@@H]1O[C@H]21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GID4 Q8IVV7 1/20 0.38
HTR2C P28335 6/20 0.34
HTR2B P41595 4/20 0.34
SLC6A2 P23975 2/20 0.33
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
KDM1A O60341 1/20 0.33
SLC6A3 Q01959 1/20 0.33
PIM1 P11309 1/20 0.32
CSNK1A1 P48729 1/20 0.32
CDK5 Q00535 1/20 0.32
ROCK1 Q13464 1/20 0.32
DYRK1A Q13627 1/20 0.32
LRRK2 Q5S007 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
BRD4 O60885 1/20 0.31
ADRA2A P08913 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26597517 1.00 KDM4E (0.40) KDM4EALDH1A1GID4HTR2CHTR2B
SCHEMBL7919137 1.00 KDM4E (0.40) KDM4EALDH1A1GID4HTR2CHTR2B
SCHEMBL18650999 0.81 GID4 (0.42) KDM4EALDH1A1GID4HTR2CHTR2B
SCHEMBL11452212 0.76 TRPM5 (0.40) HTR2CHTR2BHTR2AKDM1AADRA2A
SCHEMBL12362687 0.76 ACHE (0.38) ALDH1A1HTR2CHTR2BSLC6A2HTR2A
SCHEMBL12362682 0.76 CHRNB2 (0.44) HTR2CHTR2BHTR2AKDM1A
SCHEMBL13457936 0.76 ACHE (0.38) ALDH1A1HTR2CHTR2BSLC6A2HTR2A
SCHEMBL15021507 0.76
SCHEMBL24029486 0.73 KDM4E (0.38) KDM4EALDH1A1HTR2CHTR2BSLC6A2
SCHEMBL11104256 0.72 HTR1A (0.39) BRD4ADRA2AADRA2BADRA2CPARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3492465-B1 S1P1 AGONIST AND APPLICATION THEREOF SHIJIAZHUANG SAGACITY NEW DRUG DEV CO LTD (CN) 2021-03-24 EP disclosed
EP-3492465-A1 S1P1 AGONIST AND APPLICATION THEREOF Shijiazhuang Sagacity New Drug Development Co., Ltd. (CN) 2019-06-05 EP disclosed