Depramine

Depramine

SCHEMBL2108027

CN(C)CCCN1c2ccccc2C=Cc2ccccc21

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.73
DRD2 P14416 8/20 0.73
HRH1 P35367 8/20 0.73
HTR2A P28223 7/20 0.73
SLC6A4 P31645 7/20 0.73
HTR6 P50406 6/20 0.73
CYP2D6 P10635 8/20 0.63
CYP1A2 P05177 7/20 0.63
LMNA P02545 6/20 0.63
MAPT P10636 6/20 0.63
CHRM2 P08172 5/20 0.63
CHRM1 P11229 5/20 0.63
ADRA2B P18089 5/20 0.63
ADRA2C P18825 5/20 0.63
DRD1 P21728 5/20 0.63
SLC6A2 P23975 5/20 0.63
ADRA1A P35348 5/20 0.63
OPRM1 P35372 5/20 0.63
DRD3 P35462 5/20 0.63
KCNH2 Q12809 5/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Depramine SCHEMBL29489714 1.00 HTR1A (0.73) HTR1ADRD2HRH1HTR2ASLC6A4
Tienopramine SCHEMBL29388629 0.86 HTR1A (0.57) HTR1ADRD2HRH1HTR2ASLC6A4
SCHEMBL2525591 0.80 SLC6A4 (0.54) HTR1ADRD2HRH1HTR2ASLC6A4
SCHEMBL12265301 0.79 CYP2D6 (0.66) HTR1ADRD2HRH1HTR2ASLC6A4
SCHEMBL10613637 0.78 PTGS1 (0.53) HTR1ADRD2HRH1HTR2ASLC6A4
Promazine SCHEMBL140489 0.77 CYP2D6 (1.00) HTR1ADRD2HRH1HTR2ASLC6A4
Imipramine SCHEMBL17004048 0.77 SLC6A4 (1.00) HTR1ADRD2HRH1HTR2ASLC6A4
Imipramine SCHEMBL34282 0.77 SLC6A4 (1.00) HTR1ADRD2HRH1HTR2ASLC6A4
Promazine SCHEMBL9052694 0.77 CYP2D6 (1.00) HTR1ADRD2HRH1HTR2ASLC6A4
Imipramine SCHEMBL6118138 0.77 SLC6A4 (1.00) HTR1ADRD2HRH1HTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240307393-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT NATIONAL CANCER CENTER (KR) 2024-09-19 US claimed
EP-4368183-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT National Cancer Center (KR) 2024-05-15 EP claimed
WO-2023282544-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT 국립암센터 2023-01-12 WO claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
WO-2013126205-A1 MIXED MONOAMINE REUPTAKE INHIBITOR IN A BIODEGRADABLE POLYMER CARRIER WARSAW ORTHOPEDIC, INC. (US) 2013-08-29 WO claimed
US-20130217673-A1 MIXED MONOAMINE REUPTAKE INHIBITOR IN A BIODEGRADABLE POLYMER CARRIER WARSAW ORTHOPEDIC, INC (US) 2013-08-22 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-4249003-A Process for polycyclic amines AKTIEBOLAGET LEO (SE) 1981-02-03 US claimed
US-20240307393-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT NATIONAL CANCER CENTER (KR) 2024-09-19 US disclosed
EP-4368183-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT National Cancer Center (KR) 2024-05-15 EP disclosed
WO-2023282544-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT 국립암센터 2023-01-12 WO disclosed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed
US-20020102215-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 US disclosed
US-6331289-B1 ULTRASOUND CONTRAST AGENTS, SUSPENSION IN AQUEOUS CARRIER LIQUID OF A REPORTER COMPRISING GAS-CONTAINING OR GAS-GENERATING MATERIAL, AGENT CAPABLE OF FORMING AT LEAST TWO TYPES OF BINDING PAIRS WITH TARGET; REPORTER BEING CONJUGATED NYCOMED IMAGING AS (NO) 2001-12-18 US disclosed
US-6264917-B1 MIXTURE OF GAS FILLED MICROBUBBLES AND RELEASING AGENT NYCOMED IMAGING AS (NO) 2001-07-24 US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020102215-A1 Diagnostic/therapeutic agents BID, FUS, FABP1 HTR1A 4030/4885DRD2 4727/4885HRH1 2197/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.