SCHEMBL21088517

SCHEMBL21088517

O=C(O)c1cccc(CNC2CCCCC2)c1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPM1D O15297 3/20 0.57
POLB P06746 1/20 0.57
HDAC1 Q13547 1/20 0.54
ALDH1A1 P00352 1/20 0.54
KMO O15229 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
HIF1A Q16665 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
EPHX1 P07099 1/20 0.51
KDM1A O60341 1/20 0.51
MEP1B Q16820 1/20 0.50
CXCR4 P61073 1/20 0.50
SNCA P37840 1/20 0.49
FOLH1 Q04609 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30444177 0.92 KDM1A (0.54) PPM1DHIF1AEPHX1KDM1AMEP1B
SCHEMBL9057020 0.89 POLB (0.54) PPM1DPOLBHDAC1ALDH1A1CYP2D6
SCHEMBL791813 0.86 THRB (0.51) PPM1DHIF1AKDM1AMEP1BFOLH1
SCHEMBL15830232 0.86 PRMT5 (0.51) PPM1DKMOHIF1AKDM1AMEP1B
SCHEMBL14032272 0.84 KDM1A (0.48) PPM1DALDH1A1EPHX1KDM1AMEP1B
SCHEMBL30443983 0.82 KDM1A (0.51) PPM1DHIF1AKDM1AMEP1BFOLH1
SCHEMBL9252404 0.82 ALDH1A1 (0.68) POLBHDAC1ALDH1A1CXCR4HRH3
SCHEMBL11509945 0.82 ALDH1A1 (0.68) POLBHDAC1ALDH1A1CXCR4HRH3
SCHEMBL21089268 0.81 HDAC1 (0.72) POLBHDAC1ALDH1A1TAAR1EPHX1
SCHEMBL6911153 0.79 ALDH1A1 (0.51) POLBALDH1A1EPHX1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286172-B1 LSD1 INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS INC (US) 2019-06-12 EP disclosed