SCHEMBL21090338

SCHEMBL21090338

C/C=C\Cc1cc(C#N)c[nH]1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3285074 0.75
SCHEMBL8086280 0.72 HTR1A (0.41) HTR1ADRD2DRD4DRD3TSHR
SCHEMBL9019117 0.68 GPR84 (0.45) HTR1ADRD2DRD4DRD3TSHR
SCHEMBL4397408 0.68
SCHEMBL7505085 0.66 CYP2A6 (0.32)
SCHEMBL1779488 0.65
SCHEMBL19773472 0.64 HTR1A (0.51) HTR1ADRD2DRD4DRD3TSHR
SCHEMBL16167007 0.64 GLA (0.47)
SCHEMBL15996305 0.63
SCHEMBL8616508 0.62 LOXL2 (0.48) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019110663-A1 1,2,4-OXADIAZOLE DERIVATIVES AS HISTONE DEACETYLASE 6 INHIBITORS ORYZON GENOMICS, S.A. (ES) 2019-06-13 WO disclosed