SCHEMBL21094187

SCHEMBL21094187

CNC(O)C(C)(NC(=O)c1ccc(I)cc1)C(=O)OC

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TPMT P51580 1/20 0.37
TRPV1 Q8NER1 3/20 0.36
PLK1 P53350 1/20 0.35
MAPT P10636 2/20 0.34
HPGD P15428 1/20 0.34
GSK3B P49841 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CTSK P43235 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14714633 0.77 PLK1 (0.40) TPMTTRPV1PLK1MAPTHPGD
SCHEMBL8920815 0.72 LMNA (0.50) TPMTTRPV1MAPTHDAC1
SCHEMBL14724481 0.68 MAPK1 (0.41) MAPTGAA
SCHEMBL10938164 0.68 TRPV1 (0.33) TAS1R3TAS1R1TRPV1MAPT
SCHEMBL10938163 0.68 TRPV1 (0.33) TAS1R3TAS1R1TRPV1MAPT
SCHEMBL470103 0.68 CNR1 (0.47) TPMTTRPV1MAPTALDH1A1TDP1
SCHEMBL7807968 0.67 POLB (0.45) TAS1R3TAS1R1MAPTKDM4EALDH1A1
SCHEMBL2144483 0.66 HDAC8 (0.64) TPMTTRPV1PLK1HPGD
SCHEMBL27745010 0.66 POLB (0.47) TPMTTRPV1HDAC1
SCHEMBL7671511 0.66 CXCR2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2562155-B1 HYDROXAMIC ACID DERIVATIVE TAISHO PHARMACEUTICAL CO LTD (JP) 2019-06-05 EP disclosed