SCHEMBL21100972

SCHEMBL21100972

O=Cc1ccc(CN2CCC(CNC3CC3)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.49
KDM1A O60341 8/20 0.46
MAOB P27338 2/20 0.46
DRD2 P14416 3/20 0.45
HTR2A P28223 2/20 0.45
SLC6A4 P31645 1/20 0.45
SCN5A Q14524 1/20 0.45
HDAC6 Q9UBN7 4/20 0.44
HDAC1 Q13547 3/20 0.44
HDAC8 Q9BY41 3/20 0.44
BCHE P06276 2/20 0.44
ACHE P22303 2/20 0.44
BACE1 P56817 2/20 0.44
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21088453 0.82 DRD2 (0.50) KDM1ADRD2HTR2AHDAC6HDAC1
SCHEMBL21101096 0.81 BCHE (0.62) DRD2SLC6A4BCHEACHEBACE1
SCHEMBL20907239 0.81 ALDH1A1 (0.51) CXCR4KDM1AMAOBDRD2HTR2A
SCHEMBL28169202 0.81 CXCR4 (0.68) CXCR4KDM1AMAOBHTR2AHDAC6
SCHEMBL19725557 0.80 KDM1A (0.67) CXCR4KDM1AMAOBDRD2HTR2A
SCHEMBL21101256 0.80 SIGMAR1 (0.52) CXCR4KDM1AMAOBDRD2HTR2A
SCHEMBL21101241 0.79 ACHE (0.48) CXCR4KDM1AMAOBDRD2HTR2A
SCHEMBL21101233 0.78 SIGMAR1 (0.50) CXCR4KDM1AMAOBBCHEACHE
SCHEMBL21101338 0.78 CXCR4 (0.49) CXCR4KDM1AMAOBDRD2HTR2A
SCHEMBL23086760 0.77 DRD2 (0.48) CXCR4DRD2SLC6A4DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2688568-B1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2019-06-19 EP disclosed