SCHEMBL21153739

SCHEMBL21153739

Cc1c(CS)cccc1-c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 14/20 0.69
PDCD1 Q15116 2/20 0.69
DPP4 P27487 1/20 0.45
FOLH1 Q04609 1/20 0.45
PTGS1 P23219 1/20 0.41
EPHX1 P07099 1/20 0.41
KMT2A Q03164 1/20 0.39
IDO1 P14902 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL607544 0.82 CD274 (0.71) CD274PDCD1DPP4FOLH1PTGS1
SCHEMBL29558512 0.82 CD274 (1.00) CD274PDCD1DPP4FOLH1PTGS1
SCHEMBL358303 0.82 CD274 (1.00) CD274PDCD1DPP4FOLH1PTGS1
SCHEMBL2209528 0.81 DPP4 (0.60) CD274PDCD1DPP4FOLH1KMT2A
SCHEMBL30084702 0.80 CD274 (0.69) CD274PDCD1DPP4PTGS1EPHX1
SCHEMBL3793203 0.80 CD274 (0.69) CD274PDCD1DPP4PTGS1EPHX1
SCHEMBL7107915 0.80 CD274 (0.69) CD274PDCD1DPP4PTGS1EPHX1
SCHEMBL7194801 0.80 CD274 (0.69) CD274PDCD1DPP4FOLH1PTGS1
SCHEMBL4151221 0.80 CD274 (0.69) CD274PDCD1DPP4PTGS1EPHX1
SCHEMBL25060697 0.79 CD274 (0.62) CD274PDCD1DPP4FOLH1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113582971-B Small molecule immunosuppressant, preparation method and application thereof 北京康辰药业股份有限公司 2023-10-20 CN disclosed
CN-113582971-A Small molecule immunosuppressant, preparation method and application thereof 北京康辰药业股份有限公司 2021-11-02 CN disclosed
US-11008596-B2 Cytochrome P450 BM3 enzyme variants for preparation of cyclopropanes CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-05-18 US disclosed
US-20190211367-A1 VIVO AND IN VITRO OLEFIN CYCLOPROPANATION CATALYZED BY HEME ENZYMES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2019-07-11 US disclosed